SCHEMBL4398008

SCHEMBL4398008

COc1cc(-c2ccccc2F)cc(C2(c3ccncc3)N=C(N)c3ncccc32)c1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.43
KCNH2 Q12809 7/20 0.43
BACE2 Q9Y5Z0 6/20 0.42
CTSD P07339 5/20 0.38
TEK Q02763 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3633227 0.82 BACE1 (0.58) BACE1KCNH2BACE2CTSD
SCHEMBL3243720 0.80 BACE1 (0.48) BACE1KCNH2BACE2CTSD
SCHEMBL3992538 0.79 BACE1 (0.43) BACE1KCNH2BACE2TEK
SCHEMBL3636805 0.77 BACE1 (0.57) BACE1KCNH2BACE2CTSD
SCHEMBL3640265 0.75 BACE1 (0.65) BACE1KCNH2BACE2CTSD
SCHEMBL3633787 0.75 BACE1 (0.61) BACE1KCNH2BACE2CTSD
SCHEMBL4398010 0.74 TEK (0.36) BACE1KCNH2BACE2CTSDTEK
SCHEMBL2087395 0.73 BACE1 (0.60) BACE1KCNH2BACE2CTSD
SCHEMBL3548391 0.72 BACE1 (0.71) BACE1KCNH2BACE2CTSD
SCHEMBL3635662 0.71 BACE1 (0.58) BACE1KCNH2BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629356-B2 Substituted pyrrolo[3,4-b]pyridinamines and pharmaceutical compositions ASTRAZENECA AB (SE) 2009-12-08 US disclosed