SCHEMBL4398302

SCHEMBL4398302

Cc1c(S(=O)(=O)Nc2ccc(C#N)cc2)cc(C(=O)O)c(=O)n1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 4/20 0.55
ELANE P08246 9/20 0.51
MCL1 Q07820 2/20 0.48
NOTUM Q6P988 2/20 0.48
SLC22A12 Q96S37 1/20 0.44
CYP2C9 P11712 2/20 0.42
CPT2 P23786 1/20 0.42
CPT1A P50416 1/20 0.42
CPT1B Q92523 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8067137 0.79 ELANE (0.52) ELANENOTUMCYP2C9CYP3A4
SCHEMBL4124463 0.79 ELANE (0.63) IDH1ELANENOTUMCYP2C9CYP3A4
SCHEMBL8236829 0.78 NOTUM (0.60) ELANENOTUMCYP2C9
SCHEMBL5496689 0.78 ELANE (0.62) ELANE
SCHEMBL983524 0.77 ELANE (0.50) ELANENOTUMCYP2C9CYP3A4
SCHEMBL5490151 0.76 ELANE (0.62) ELANE
SCHEMBL4123923 0.76 ELANE (0.51) ELANECYP2C9CYP3A4
SCHEMBL29808797 0.75 NOTUM (0.76) ELANENOTUM
SCHEMBL5752612 0.75 NOTUM (0.76) ELANENOTUM
SCHEMBL4131190 0.75 ELANE (0.68) ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2064184-A1 MULTIMERIC HETEROCYCLIC COMPOUNDS USEFUL AS NEUTROPHIL ELASTASE INHIBITORS AstraZeneca AB (SE) 2009-06-03 EP disclosed
WO-2008030158-A1 MULTIMERIC HETEROCYCLIC COMPOUNDS USEFUL AS NEUTROPHIL ELASTASE INHIBITORS ASTRAZENECA AB (SE) 2008-03-13 WO disclosed