SCHEMBL4398964

SCHEMBL4398964

NN=C(N)c1ccc2[nH]ccc2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.64
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
MAPT P10636 1/20 0.56
CYP2C19 P33261 1/20 0.56
RAB9A P51151 1/20 0.56
USP2 O75604 1/20 0.48
GAA P10253 1/20 0.48
ALOX15 P16050 1/20 0.48
RAD51 Q06609 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
CTNNB1 P35222 3/20 0.46
WNT3A P56704 3/20 0.46
GRIN2D O15399 1/20 0.45
GRIN3B O60391 1/20 0.45
GRIN1 Q05586 1/20 0.45
GRIN2A Q12879 1/20 0.45
GRIN2B Q13224 1/20 0.45
GRIN2C Q14957 1/20 0.45
GRIN3A Q8TCU5 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4403840 0.98 F2 (0.62) F2CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL2416081 0.86 CYP1A2 (0.65) F2CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL403839 0.86 CYP1A2 (0.65) F2CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL27522161 0.78 F2 (0.68) F2CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL563181 0.78 F2 (1.00) F2CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL170646 0.78 F2 (0.68) F2CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL29858415 0.78 F2 (0.68) F2CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL3708430 0.78 F2 (0.68) F2CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL29540009 0.78 F2 (0.68) F2CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL28604703 0.77 MAPT (0.54) F2CYP1A2CYP3A4MAPTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101321525-B Heteroaryl substituted piperidine derivatives as L-CPT1 inhibitors HOFFMANN LA ROCHE 2013-01-30 CN disclosed
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed