SCHEMBL4399223

SCHEMBL4399223

ON=C(Cl)c1cncc(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.55
SMYD3 Q9H7B4 1/20 0.38
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4399222 1.00 HCAR2 (0.55) HCAR2SMYD3MKNK1MKNK2CHRNB4
SCHEMBL14395549 0.79 HCAR2 (0.52) HCAR2SMYD3MKNK1MKNK2
SCHEMBL14755489 0.79 HCAR2 (0.52) HCAR2SMYD3MKNK1MKNK2CHRNB4
SCHEMBL4392022 0.77 HCAR2 (0.53) HCAR2
SCHEMBL4392027 0.77 HCAR2 (0.53) HCAR2
SCHEMBL14183649 0.77 TPMT (0.44)
SCHEMBL15635597 0.77 TPMT (0.44)
SCHEMBL12818742 0.77 TPMT (0.44)
SCHEMBL4196968 0.76 HCAR2 (0.69) HCAR2SMYD3MKNK1MKNK2PKM
SCHEMBL28835397 0.75 HCAR2 (0.57) HCAR2MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8383658-B2 Isoxazole based neuronal nicotinic receptor ligands and methods of use ABBOTT LABORATORIES (US) 2013-02-26 US disclosed
US-20090306096-A1 Novel Isoxazoles and Methods of Use Thereof ABBOTT LABORATORIES (US) 2009-12-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090306096-A1 Novel Isoxazoles and Methods of Use Thereof XDH, PRDX5, CYP4X1 HCAR2 672/4885SMYD3 3778/4885MKNK1 3216/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.