SCHEMBL4400634

SCHEMBL4400634

C=CCOC(=O)C(=O)O.[Ti]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.42
MAPT P10636 4/20 0.39
TSHR P16473 2/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
ALDH1A1 P00352 5/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PKM P14618 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PTP4A3 O75365 1/20 0.33
PTP4A1 Q93096 1/20 0.33
SNCA P37840 1/20 0.33
APP P05067 1/20 0.33
KDM4E B2RXH2 1/20 0.32
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669729 0.97
SCHEMBL3458279 0.95 CYP3A4 (0.42) CYP3A4MAPTTSHRCACNA1BAPBA1
Hydrochloric Acid SCHEMBL9595329 0.95 CYP3A4 (0.42) CYP3A4MAPTTSHRCACNA1BAPBA1
SCHEMBL177943 0.84 CYP3A4 (0.48) CYP3A4MAPTTSHRCACNA1BAPBA1
SCHEMBL10497073 0.83 CYP3A4 (0.35) CYP3A4MAPTTSHRCACNA1BAPBA1
SCHEMBL7512684 0.81 CYP3A4 (0.46) CYP3A4MAPTTSHRCACNA1BAPBA1
SCHEMBL11277855 0.81 CYP3A4 (0.39) CYP3A4MAPTTSHRCACNA1BAPBA1
SCHEMBL11278938 0.81 CYP3A4 (0.39) CYP3A4MAPTTSHRCACNA1BAPBA1
SCHEMBL2733016 0.81 CYP3A4 (0.39) CYP3A4MAPTTSHRCACNA1BAPBA1
SCHEMBL44692 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805243-B1 POLYTRIMETHYLENE TEREPHTHALATE HAVING A LOW LEVEL OF ACROLEIN AND A PROCESS FOR PRODUCING THE SAME LURGI ZIMMER GMBH (DE) 2013-01-09 EP disclosed
US-20120141723-A1 POLYMER FIBER CONTAINING FLAME RETARDANT, PROCESS FOR PRODUCING THE SAME, AND MATERIAL CONTAINING SUCH FIBERS SHELL OIL COMPANY 2012-06-07 US disclosed
EP-2084170-A1 POLYMER FIBER CONTAINING FLAME RETARDANT, PROCESS FOR PRODUCING THE SAME, AND MATERIAL CONTAINING SUCH FIBERS Shell Internationale Research Maatschappij B.V. (NL) 2009-08-05 EP disclosed
EP-2084169-A1 POLYMER COMPOSITION CONTAINING FLAME RETARDANT AND PROCESS FOR PRODUCING THE SAME Shell Internationale Research Maatschappij B.V. (NL) 2009-08-05 EP disclosed
US-20080194793-A1 POLYTRIMETHYLENE TEREPHTHALATE HAVING A LOW LEVEL OF ACROLEIN AND A PROCESS FOR PRODUCING THE SAME KELSEY DONALD ROSS 2008-08-14 US disclosed
US-20080132620-A1 POLYMER COMPOSITION CONTAINING FLAME RETARDANT AND PROCESS FOR PRODUCING THE SAME SHELL OIL COMPANY 2008-06-05 US disclosed
US-7381787-B2 Polytrimethylene terephthalate having a low level of acrolein and a process for producing the same SHELL OIL COMPANY (US) 2008-06-03 US disclosed
WO-2008061075-A1 POLYMER COMPOSITION CONTAINING FLAME RETARDANT AND PROCESS FOR PRODUCING THE SAME SHELL OIL COMPANY (US) 2008-05-22 WO disclosed
WO-2008061087-A1 POLYMER FIBER CONTAINING FLAME RETARDANT, PROCESS FOR PRODUCING THE SAME, AND MATERIAL CONTAINING SUCH FIBERS SHELL OIL COMPANY (US) 2008-05-22 WO disclosed
EP-1805243-A1 POLYTRIMETHYLENE TEREPHTHALATE HAVING A LOW LEVEL OF ACROLEIN AND A PROCESS FOR PRODUCING THE SAME SHELL INTERNATIONAL RESEARCH MAATSCHAPPIJ B.V. (NL) 2007-07-11 EP disclosed
US-20060084783-A1 Polytrimethylene terephthalate having a low level of acrolein and a process for producing the same LURGI ZIMMER GMBH (DE) 2006-04-20 US disclosed
WO-2006033917-A1 POLYTRIMETHYLENE TEREPHTHALATE HAVING A LOW LEVEL OF ACROLEIN AND A PROCESS FOR PRODUCING THE SAME SHELL INTERNATIONAL RESEARCH MAATSCHAPPIJ B.V. (NL) 2006-03-30 WO disclosed