SCHEMBL4401417

SCHEMBL4401417

Cc1ccc(S(=O)(=O)OC[C@@H]2CCCN(C(=O)O)C2C(C)(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
POLB P06746 2/20 0.40
CYP2D6 P10635 2/20 0.39
STAT3 P40763 1/20 0.37
KDM4E B2RXH2 2/20 0.37
CYP1A2 P05177 1/20 0.37
MAPK1 P28482 1/20 0.37
ATM Q13315 1/20 0.37
GAA P10253 2/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
FFAR1 O14842 1/20 0.36
TSHR P16473 1/20 0.36
ACHE P22303 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16823465 1.00 ALDH1A1 (0.40) ALDH1A1POLBCYP2D6STAT3KDM4E
SCHEMBL14994148 0.93 CYP2D6 (0.40) ALDH1A1POLBCYP2D6STAT3KDM4E
SCHEMBL14994147 0.93 CYP2D6 (0.40) ALDH1A1POLBCYP2D6STAT3KDM4E
SCHEMBL14995618 0.87 STAT3 (0.39) ALDH1A1POLBCYP2D6STAT3CYP1A2
SCHEMBL505551 0.87 CYP2D6 (0.37) ALDH1A1POLBCYP2D6STAT3KDM4E
SCHEMBL26117855 0.83 ALDH1A1 (0.46) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2302585 0.83 FFAR1 (0.45) ALDH1A1POLBCYP2D6STAT3KDM4E
SCHEMBL3129424 0.83 FFAR1 (0.45) ALDH1A1POLBCYP2D6STAT3KDM4E
SCHEMBL3616703 0.83 FFAR1 (0.45) ALDH1A1POLBCYP2D6STAT3KDM4E
SCHEMBL18173559 0.83 CYP2D6 (0.48) ALDH1A1POLBCYP2D6KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924572-B1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SMITHKLINE BEECHAM CORP (US) 2009-12-30 EP disclosed