SCHEMBL4402298

SCHEMBL4402298

CCOC(=O)c1cncc(C(=O)NO)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.69
CYP2C9 P11712 1/20 0.69
SMN1; SMN2 Q16637 3/20 0.55
ALDH1A1 P00352 3/20 0.52
MAPT P10636 1/20 0.52
POLB P06746 1/20 0.52
TSHR P16473 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
HSD17B10 Q99714 1/20 0.52
KMT2A Q03164 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
ATM Q13315 1/20 0.47
KDM4E B2RXH2 2/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL277284 0.88 CYP2C19 (0.86) CYP2C19CYP2C9SMN1; SMN2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL9679507 0.86 CYP2C19 (0.83) CYP2C19CYP2C9SMN1; SMN2ALDH1A1MAPT
SCHEMBL28328600 0.85 CYP2C19 (0.75) CYP2C19CYP2C9SMN1; SMN2ALDH1A1MAPT
SCHEMBL5485762 0.84 CA12 (0.58) CYP2C19CYP2C9SMN1; SMN2ALDH1A1MAPT
SCHEMBL4405655 0.84 CYP2C19 (0.65) CYP2C19CYP2C9SMN1; SMN2ALDH1A1MAPT
SCHEMBL158686 0.81 CYP2C19 (0.70) CYP2C19CYP2C9SMN1; SMN2MAPTPOLB
SCHEMBL2112657 0.81 CYP2C19 (1.00) CYP2C19CYP2C9SMN1; SMN2ALDH1A1MAPT
SCHEMBL29597594 0.81 CYP2C19 (0.70) CYP2C19CYP2C9SMN1; SMN2MAPTPOLB
Hydrochloric Acid SCHEMBL3334480 0.80 CYP2C19 (0.73) CYP2C19CYP2C9SMN1; SMN2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL3336664 0.80 CYP2C19 (0.97) CYP2C19CYP2C9SMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed