SCHEMBL277284

SCHEMBL277284

CCOC(=O)c1cncc(C(=O)OCC)c1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.86
CYP2C9 P11712 1/20 0.86
CA12 O43570 3/20 0.57
CA1 P00915 3/20 0.57
CA2 P00918 3/20 0.57
CA7 P43166 3/20 0.57
CA9 Q16790 3/20 0.57
CA14 Q9ULX7 3/20 0.57
ALDH1A1 P00352 1/20 0.54
MAPT P10636 1/20 0.54
ATM Q13315 1/20 0.53
ESR1 P03372 1/20 0.52
ESR2 Q92731 1/20 0.52
CYP1A2 P05177 3/20 0.50
CYP3A4 P08684 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
LMNA P02545 1/20 0.50
MAOA P21397 1/20 0.50
KMT2A Q03164 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9679507 0.98 CYP2C19 (0.83) CYP2C19CYP2C9CA12CA1CA2
SCHEMBL2112657 0.93 CYP2C19 (1.00) CYP2C19CYP2C9CA12CA1CA2
SCHEMBL28328600 0.93 CYP2C19 (0.75) CYP2C19CYP2C9CA12CA1CA2
Hydrochloric Acid SCHEMBL3334480 0.91 CYP2C19 (0.73) CYP2C19CYP2C9CA12CA1CA2
Hydrochloric Acid SCHEMBL3336664 0.91 CYP2C19 (0.97) CYP2C19CYP2C9CA12CA1CA2
SCHEMBL6979199 0.90 CYP2C19 (0.72) CYP2C19CYP2C9CA12CA1CA2
Potassium Ion SCHEMBL28014022 0.89 CYP2C19 (0.71) CYP2C19CYP2C9CA12CA1CA2
SCHEMBL158686 0.89 CYP2C19 (0.70) CYP2C19CYP2C9MAPTATMCYP1A2
SCHEMBL29597594 0.89 CYP2C19 (0.70) CYP2C19CYP2C9MAPTATMCYP1A2
SCHEMBL1812268 0.89 CYP2C9 (0.70) CYP2C19CYP2C9CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939568-A Accelerated catalysis of olefinic epoxidations THE SCRIPPS RESEARCH INSTITUTE (US) 1999-08-17 US claimed
CN-117534684-A pan-KRAS inhibitor compound 杭州阿诺生物医药科技有限公司 2024-02-09 CN disclosed
US-20230295125-A1 METALLOENZYME INHIBITORS FOR TREATING CANCERS, ALZHEIMER'S DISEASE, HEMOCHROMATOSIS, AND OTHER DISORDERS MIRALOGX LLC (US) 2023-09-21 US disclosed
US-20230295125-A1 METALLOENZYME INHIBITORS FOR TREATING CANCERS, ALZHEIMER'S DISEASE, HEMOCHROMATOSIS, AND OTHER DISORDERS MIRALOGX LLC (US) 2023-09-21 US disclosed
WO-2022138888-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF 東レ株式会社 2022-06-30 WO disclosed
WO-2022082079-A1 METALLOENZYME INHIBITORS FOR TREATING CANCERS, ALZHEIMER'S DISEASE, HEMOCHROMATOSIS, AND OTHER DISORDERS METALLO THERAPIES, INC. (US) 2022-04-21 WO disclosed
CN-114133329-A Cis-configuration 2, 2-difluoro-4-phenylbutan-3-ethyl enoate compound and preparation method thereof 上海大学 2022-03-04 CN disclosed
EP-2360161-B1 Preparation and use of magnesium amides MUNICHEM GMBH (DE) 2016-08-31 EP disclosed
WO-2016120635-A1 PROCESSES FOR THE PREPARATION OF COMPOUNDS, SUCH AS 3-ARYLBUTANALS, USEFUL IN THE SYNTHESIS OF MEDETOMIDINE CAMBREX KARLSKOGA AB (SE) 2016-08-04 WO disclosed
US-8134005-B2 Preparation and use of magnesium amides Ludwig-Maximilians-Universitat München (DE) 2012-03-13 US disclosed
US-4968803-A FLUORINE AS OXIDANT ALLIED-SIGNAL INC. (US) 1990-11-06 US disclosed
US-4900837-A Brain-specific drug delivery of steroid sex hormones cleaved from pyridinium carboxylates and dihydro-pyridine carboxylate precursors UNIVERSITY OF FLORIDA (US) 1990-02-13 US disclosed
US-4880921-A Brain-specific drug delivery UNIVERSITY OF FLORIDA (US) 1989-11-14 US disclosed
US-4824850-A DIHYDROPYRIDINE-PYRIDINIUM SALT REDOX CARRIER UNIVERSITY OF FLORIDA (US) 1989-04-25 US disclosed
EP-0267794-A2 Process for preparing polyolefins Nippon Petrochemicals Co., Ltd. (JP) 1988-05-18 EP disclosed
EP-0194752-A1 Dihydropyridine alkanol amines, process for their preparation and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-09-17 EP disclosed
US-4540564-A DIHYDROPYRIDINE AND/OR PYRIDINIUM SALT REDOX CARRIER UNIVERSITY OF FLORIDA (US) 1985-09-10 US disclosed
US-4525555-A TITANIUM COMPOUND SUPPORTED ON SOLID REACTION PRODUCT OF MAGNESIUM HALIDE, SILOXANES, ORGANIC COMPOUNDS NIPPON OIL COMPANY, LIMITED (JP) 1985-06-25 US disclosed
EP-0110955-A1 BRAIN-SPECIFIC DRUG DELIVERY. UNIV FLORIDA (US) 1984-06-20 EP disclosed
WO-1983003968-A1 BRAIN-SPECIFIC DRUG DELIVERY UNIVERSITY OF FLORIDA (US) 1983-11-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230295125-A1 METALLOENZYME INHIBITORS FOR TREATING CANCERS, ALZHEIMER'S DISEASE, HEMOCHROMATOSIS, AND OTHER DISORDERS HMOX1, FECH, SLC40A1 CYP2C19 375/4885CYP2C9 689/4885CA12 1042/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.