SCHEMBL4403750

SCHEMBL4403750

Cc1cc[n+](CCCc2cccc(CCC[n+]3ccc(C)cc3C)c2)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.41
NPC1 O15118 2/20 0.40
POLB P06746 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CHRNA7 P36544 2/20 0.36
CHRNA10 Q9GZZ6 2/20 0.36
CHRNA9 Q9UGM1 2/20 0.36
HRH3 Q9Y5N1 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
NOS1 P29475 4/20 0.34
NOS2 P35228 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
NOS3 P29474 2/20 0.33
IDO1 P14902 1/20 0.33
FDPS P14324 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4400673 0.94 NPC1 (0.45) TAAR1NPC1POLBRAB9ASMN1; SMN2
SCHEMBL4401493 0.85 CHRNA7 (0.46) NPC1POLBRAB9ASMN1; SMN2CHRNA7
SCHEMBL13334053 0.84 NPC1 (0.49) NPC1POLBRAB9ASMN1; SMN2CHRNA7
SCHEMBL4400594 0.83 NPC1 (0.42) NPC1POLBRAB9ASMN1; SMN2CHRNA7
Bromide SCHEMBL3317318 0.83 NPC1 (0.51) NPC1POLBRAB9ASMN1; SMN2CHRNA7
SCHEMBL8015063 0.82 NPC1 (0.45) NPC1POLBRAB9ASMN1; SMN2KDM4E
SCHEMBL4404758 0.81 NPC1 (0.44) NPC1POLBRAB9ASMN1; SMN2CHRNA7
SCHEMBL4404565 0.81 NPC1 (0.62) TAAR1NPC1POLBRAB9ASMN1; SMN2
Bromide SCHEMBL7251134 0.80 NPC1 (0.48) NPC1POLBRAB9ASMN1; SMN2KDM4E
SCHEMBL13334261 0.79 CHRNA7 (0.46) NPC1POLBRAB9ASMN1; SMN2CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178678-B2 Bis-quaternary ammonium salts and methods for modulating neuronal nicotinic acetylcholine receptors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2012-05-15 US disclosed
US-20100069432-A1 Bis-Quaternary Ammonium Salts and Methods for Modulating Neuronal Nicotinic Acetylcholine Receptors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2010-03-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069432-A1 Bis-Quaternary Ammonium Salts and Methods for Modulating Neuronal Nicotinic Acetylcholine Receptors CHRNA2, CHRNA5, CHRNA4 TAAR1 55/4885NPC1 1844/4885POLB 3604/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.