SCHEMBL4403769

SCHEMBL4403769

COc1cc(C(C)=O)cc2c(C)n[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.49
ADORA2A P29274 2/20 0.36
ADORA2B P29275 2/20 0.36
CNR2 P34972 1/20 0.36
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP3A4 P08684 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA3 P07451 1/20 0.34
PKM P14618 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA7 P43166 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1144821 0.88 CNR2 (0.49) LMNACNR2KMT2ATSHRCA12
SCHEMBL16167682 0.84 LMNA (0.35) LMNAADORA2AADORA2BCNR2KMT2A
SCHEMBL1144834 0.83 HSD17B2 (0.49) LMNAKMT2ASMN1; SMN2TSHRCA12
SCHEMBL4402971 0.82 ADORA2A (0.41) LMNAADORA2AADORA2BKMT2ASMN1; SMN2
SCHEMBL31637404 0.72 TSHR (0.44) LMNACYP2C9TSHRCYP2C19ALDH1A1
SCHEMBL31637418 0.72 PDE4D (0.45) KMT2ASMN1; SMN2CYP2C9CYP2C19CA12
SCHEMBL12327904 0.70 LMNA (0.69) LMNACNR2KMT2ACYP3A4CYP1A2
SCHEMBL1145074 0.70 HSD17B2 (0.47) LMNAKMT2ASMN1; SMN2TSHRCA12
SCHEMBL1144379 0.70 CA12 (0.45) CNR2KMT2ATSHRCA12CA1
SCHEMBL1145053 0.69 ADORA2A (0.41) LMNAADORA2AADORA2BKMT2ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012056372-A1 N1/N2-LACTAM ACETYL-CoA CARBOXYLASE INHIBITORS PFIZER INC. (US) 2012-05-03 WO disclosed