SCHEMBL4404077

SCHEMBL4404077

O=C(c1nccc2ccccc12)c1nccc2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.64
RAB9A P51151 2/20 0.54
PLAU P00749 2/20 0.50
CYP2A6 P11509 1/20 0.50
F12 P00748 1/20 0.50
NCF1 P14598 1/20 0.50
NOS3 P29474 1/20 0.50
NOS1 P29475 1/20 0.50
NOS2 P35228 1/20 0.50
BACE1 P56817 1/20 0.50
MAPT P10636 2/20 0.47
TSHR P16473 2/20 0.47
MEN1 O00255 1/20 0.47
TP53 P04637 1/20 0.47
KMT2A Q03164 1/20 0.47
PLG P00747 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31357187 0.89 CNR2 (0.70) CNR2RAB9APLAUCYP2A6F12
SCHEMBL5084291 0.89 CNR2 (0.70) CNR2RAB9APLAUCYP2A6F12
Water SCHEMBL27550989 0.87 CNR2 (0.68) CNR2RAB9APLAUCYP2A6F12
SCHEMBL13475588 0.87 CNR2 (0.68) CNR2RAB9AMAPTMEN1KMT2A
Silver SCHEMBL11452821 0.86 CNR2 (0.55) CNR2RAB9APLAUCYP2A6F12
SCHEMBL28091074 0.86 CNR2 (0.55) CNR2RAB9APLAUCYP2A6F12
Lithium Ion SCHEMBL29972760 0.86 CNR2 (0.55) CNR2RAB9APLAUCYP2A6F12
SCHEMBL287165 0.86 RAB9A (0.56) CNR2RAB9APLAUCYP2A6F12
SCHEMBL5357601 0.86 CNR2 (0.54) CNR2RAB9APLAUCYP2A6F12
SCHEMBL13475580 0.86 CNR2 (0.55) CNR2RAB9AMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 119 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110041257-B Method for synthesizing indene spiro indene [1,2-c ] isoquinoline triketone compound 河南师范大学 2021-08-03 CN claimed
CN-110105359-B Method for synthesizing indene spiro isoindole [2,1-b ] isoquinoline triketone compound 河南师范大学 2021-08-03 CN claimed
CN-108997339-B Method for synthesizing isoindole [2,1-b ] isoquinoline-7-carboxylic ester compound 河南师范大学 2021-01-29 CN claimed
CN-110305062-A Substituted isoquinoline ketone compounds and its synthetic method and application 广州医科大学 2019-10-08 CN claimed
CN-110183379-A A kind of copper catalysis one kettle way prepares the synthetic method and application of C-4 sulfuryl substituted isoquinoline ketone compounds 青岛科技大学 2019-08-30 CN claimed
CN-109734662-A A kind of trifluoromethyl substituted-dihydro isoquinolinone derivatives and preparation method thereof 郑州大学 2019-05-10 CN claimed
CN-108997339-A A method of synthesis iso-indoles [2,1-b] isoquinolin -7- carboxylic acid ester compound 河南师范大学 2018-12-14 CN claimed
CN-107021958-A FXR receptor stimulating agents 山东轩竹医药科技有限公司 2017-08-08 CN claimed
CN-106674109-A Method for synthesizing anti-cancer inhibitor intermediate 温州医科大学附属第二医院 2017-05-17 CN claimed
CN-105859617-A Fluoroisoquinolone compound and synthesis method thereof 叶芳 2016-08-17 CN claimed
CN-103025383-A Compounds for the treatment of clostridium difficile-associated diseases SUMMIT CORP PLC 2013-04-03 CN claimed
CN-100558728-C Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2009-11-11 CN claimed
CN-1972929-A Heterocyclic CGRP antagonists for the treatment of migraine BRISTOL MYERS SQUIBB CO (US) 2007-05-30 CN claimed
CN-1671711-A Calcitonin gene related peptide receptor antagonists BRISTOL MYERS SQUIBB CO (US) 2005-09-21 CN claimed
CN-115260096-B Method for synthesizing dihydroisoquinolinones based on carbon monoxide gas or carbon monoxide substitution source 武汉大学 2024-04-09 CN disclosed
CN-115260096-B Method for synthesizing dihydroisoquinolinones based on carbon monoxide gas or carbon monoxide substitution source 武汉大学 2024-04-09 CN disclosed
CN-113748104-B Isoquinolinones for inhibiting SSAO/VAP-1 and application thereof 广东东阳光药业股份有限公司 2024-02-27 CN disclosed
CN-1520296-A Amino nicotinate derivatives as glucokinase (GLK) modulators 2004-08-11 CN disclosed
CN-1449443-A Fungal cell wall synthetic genes EISAI CO LTD (JP) 2003-10-15 CN disclosed
EP-1300464-A1 FUNGAL CELL WALL SYNTHESIS GENE Eisai Co., Ltd. (JP) 2003-04-09 EP disclosed