SCHEMBL4407857

SCHEMBL4407857

CSc1sc(C(=O)N2CCC(c3cccc(CN)c3)CC2)c2c1C=CCC2

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
KCNH2 Q12809 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
TPSAB1 Q15661 9/20 0.47
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1382133 0.94 TPSAB1 (0.52) TPSAB1
SCHEMBL4403180 0.81 CYP3A4 (0.49) CYP3A4CYP2D6KCNH2TPSAB1KDM4E
Trifluoroacetic Acid SCHEMBL1382520 0.77 TPSAB1 (0.52) TPSAB1
SCHEMBL18652756 0.76 CYP3A4 (0.49) CYP3A4CYP2D6KCNH2TPSAB1
SCHEMBL18652812 0.76 CYP3A4 (0.49) CYP3A4CYP2D6KCNH2TPSAB1
SCHEMBL15788518 0.76 CYP3A4 (0.49) CYP3A4CYP2D6KCNH2TPSAB1
SCHEMBL15788517 0.76 CYP3A4 (0.49) CYP3A4CYP2D6KCNH2TPSAB1
SCHEMBL4404783 0.74 CYP3A4 (0.47) CYP3A4CYP2D6KCNH2TPSAB1
SCHEMBL15866752 0.74 CYP3A4 (0.55) CYP3A4CYP2D6KCNH2TPSAB1
Trifluoroacetic Acid SCHEMBL6317047 0.74 TPSAB1 (0.51) TPSAB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296972-B1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS AVENTIS PHARMA INC (US) 2009-12-23 EP claimed