SCHEMBL4411155

SCHEMBL4411155

Cn1cc(-c2ccccc2)c2ccc(C(=O)[C@@H]3C(=O)c4cc(-c5nnn[nH]5)ccc4OC34CCNCC4)cc21

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 8/20 0.37
BRD4 O60885 1/20 0.31
SCN5A Q14524 2/20 0.31
OPRD1 P41143 2/20 0.31
CYP2D6 P10635 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4417848 0.85 KHK (0.38)
SCHEMBL4414233 0.82 HPGD (0.32)
SCHEMBL4427903 0.82 KHK (0.35) OPRD1CYP2D6KCNH2
SCHEMBL4267712 0.80 OPRD1 (0.32) OPRD1CYP2D6KCNH2
SCHEMBL4266728 0.80 OPRD1 (0.32) OPRD1CYP2D6KCNH2
SCHEMBL4266808 0.80 OPRD1 (0.32) OPRD1CYP2D6KCNH2
SCHEMBL4418733 0.78 CRBN (0.36)
SCHEMBL733137 0.77 HDAC3 (0.47)
SCHEMBL4883777 0.77
SCHEMBL4270727 0.77 PIP5K1C (0.32) BRD4OPRD1CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP disclosed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO disclosed