SCHEMBL4412807

SCHEMBL4412807

NCc1cccc(C2CCN(C(=O)c3cccc(C#Cc4ccccc4F)c3)CC2)c1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 11/20 0.50
F10 P00742 1/20 0.47
TACR2 P21452 1/20 0.45
TACR1 P25103 1/20 0.45
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1382400 0.95 TPSAB1 (0.58) TPSAB1F10
Hydrochloric Acid SCHEMBL4399035 0.88 TPSAB1 (0.54) TPSAB1F10CYP3A4CYP2D6KCNH2
Trifluoroacetic Acid SCHEMBL4408071 0.85 TPSAB1 (0.59) TPSAB1F10
Trifluoroacetic Acid SCHEMBL4398566 0.85 TPSAB1 (0.55) TPSAB1F10
Trifluoroacetic Acid SCHEMBL4407733 0.85 TPSAB1 (0.55) TPSAB1F10
Trifluoroacetic Acid SCHEMBL4406887 0.84 TPSAB1 (0.57) TPSAB1F10
Hydrochloric Acid SCHEMBL4406935 0.83 TPSAB1 (0.48) TPSAB1F10CYP3A4CYP2D6KCNH2
Trifluoroacetic Acid SCHEMBL4409362 0.83 TPSAB1 (0.56) TPSAB1F10
SCHEMBL301845 0.83 F10 (0.67) TPSAB1F10
Trifluoroacetic Acid SCHEMBL4411518 0.80 TPSAB1 (0.55) TPSAB1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296972-B1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS AVENTIS PHARMA INC (US) 2009-12-23 EP claimed
US-6977263-B2 Chemical compounds AVENTIS PHARMACEUTICALS INC. (US) 2005-12-20 US disclosed