SCHEMBL4413437

SCHEMBL4413437

CC1(C)CC(N2C(=O)CCC2=O)CC(C)(C)N1O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
PKM P14618 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 2/20 0.31
MAPK1 P28482 1/20 0.30
MEN1 O00255 1/20 0.30
TSHR P16473 1/20 0.30
ENO1 P06733 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13328952 0.88 GAA (0.38) GAAL3MBTL1KDM4EALDH1A1ALOX15
SCHEMBL5701242 0.82 MAPK1 (0.31) MAPK1
Bicarbonate SCHEMBL15320130 0.79 MAPK1 (0.32) MAPK1
SCHEMBL1815774 0.78 GAA (0.36) GAAL3MBTL1KDM4EALDH1A1ALOX15
SCHEMBL10577056 0.77 MAPK1 (0.32) MAPK1
SCHEMBL12301403 0.77 GAA (0.32) GAAL3MBTL1KDM4EALDH1A1ALOX15
SCHEMBL13297945 0.74 BRD4 (0.34) PKMKMT2AMEN1
SCHEMBL20850264 0.74 ALDH1A1 (0.36) GAAL3MBTL1KDM4EALDH1A1ALOX15
SCHEMBL989503 0.73 MAPK1 (0.53) GAAKDM4EALDH1A1KMT2AMAPK1
SCHEMBL16161446 0.72 GAA (0.38) GAAL3MBTL1KDM4EALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095006-A1 DERIVATIVES OF 1-OXYL-4-HYDROXY-OR 4-AMINO-2,2,6,6-TETRAMETHYLPIPERIDINE AS POLYMERIZATION INHIBITORS FOR (METH) ACRYLATE MONOMERS Ciba SC Holding AG (CH) 2001-05-02 EP claimed
WO-2000003965-A1 DERIVATIVES OF 1-OXYL-4-HYDROXY- OR 4-AMINO-2,2,6,6-TETRAMETHYLPIPERIDINE AS POLYMERIZATION INHIBITORS FOR (METH)ACRYLATE MONOMERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2000-01-27 WO claimed
US-5928558-A STORAGE STABILITY CIBA SPECIALTY CHEMICALS CORPORATION (US) 1999-07-27 US claimed
US-5006577-A Durable, weatherproof CIBA-GEIGY CORPORATION (US) 1991-04-09 US claimed
US-20210254056-A1 IDENTIFICATION AND TARGETED MODULATION OF GENE SIGNALING NETWORKS CAMP4 THERAPEUTICS CORPORATION 2021-08-19 US disclosed
US-20190192691-A1 REGULATED BIOCIRCUIT SYSTEMS OBSIDIAN THERAPEUTICS, INC. 2019-06-27 US disclosed
EP-2030963-A2 Derivatives of 1-oxyl-4-hydroxy-or 4-amino-2,2,6,6-tetramethylpiperidine as polymerization inhibitors for (meth) acrylate monomers Ciba Holding Inc. (CH) 2009-03-04 EP disclosed
US-20070072965-A1 Color fast polyurethanes CIBA SPECIALTY CHEMICALS CORPORATION 2007-03-29 US disclosed
EP-0309401-B2 Stabilization of coatings with N-hydroxy hindered amines CIBA SC HOLDING AG (CH) 2002-06-05 EP disclosed
EP-1095006-A1 DERIVATIVES OF 1-OXYL-4-HYDROXY-OR 4-AMINO-2,2,6,6-TETRAMETHYLPIPERIDINE AS POLYMERIZATION INHIBITORS FOR (METH) ACRYLATE MONOMERS Ciba SC Holding AG (CH) 2001-05-02 EP disclosed
EP-1000032-A1 INHIBITION OF PULP AND PAPER YELLOWING USING NITROXIDES AND OTHER COADDITIVES Ciba SC Holding AG (CH) 2000-05-17 EP disclosed
WO-2000003965-A1 DERIVATIVES OF 1-OXYL-4-HYDROXY- OR 4-AMINO-2,2,6,6-TETRAMETHYLPIPERIDINE AS POLYMERIZATION INHIBITORS FOR (METH)ACRYLATE MONOMERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2000-01-27 WO disclosed
WO-1999005108-A1 INHIBITION OF PULP AND PAPER YELLOWING USING NITROXIDES AND OTHER COADDITIVES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1999-02-04 WO disclosed
EP-0309401-B1 Stabilization of coatings with N-hydroxy hindered amines CIBA GEIGY AG (CH) 1994-10-26 EP disclosed
US-5064883-A Stabilization of acid catalyzed thermoset resins with n-hydroxy hindered amines CIBA-GEIGY CORPORATION (US) 1991-11-12 US disclosed
US-5006577-A Durable, weatherproof CIBA-GEIGY CORPORATION (US) 1991-04-09 US disclosed
US-5004770-A Light, heat, and oxygen resistant CIBA-GEIGY CORPORATION (US) 1991-04-02 US disclosed
EP-0309401-A1 Stabilization of coatings with N-hydroxy hindered amines CIBA-GEIGY AG (CH) 1989-03-29 EP disclosed