Etanidazole

Etanidazole

SCHEMBL4414

O=C(Cn1ccnc1[N+](=O)[O-])NCCO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 1.00
THRB P10828 1/20 1.00
CYP2C19 P33261 1/20 1.00
CYP3A4 P08684 1/20 0.65
CYP2D6 P10635 1/20 0.65
OPRK1 P41145 1/20 0.65
CA12 O43570 5/20 0.63
CA1 P00915 5/20 0.63
CA2 P00918 5/20 0.63
CA9 Q16790 5/20 0.63
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 2/20 0.43
TYMP P19971 3/20 0.40
GRIN2B Q13224 1/20 0.40
NOS1 P29475 1/20 0.38
TAAR1 Q96RJ0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Etanidazole SCHEMBL8171462 1.00 LMNA (1.00) LMNATHRBCYP2C19CYP3A4CYP2D6
Etanidazole SCHEMBL9473771 0.99 LMNA (0.97) LMNATHRBCYP2C19CYP3A4CYP2D6
Etanidazole SCHEMBL27849456 0.95 LMNA (0.90) LMNATHRBCYP2C19CYP3A4CYP2D6
Etanidazole SCHEMBL16246698 0.94 LMNA (0.88) LMNATHRBCYP2C19CYP3A4CYP2D6
Etanidazole SCHEMBL28152496 0.94 LMNA (0.88) LMNATHRBCYP2C19CYP3A4CYP2D6
Etanidazole SCHEMBL7915363 0.89 LMNA (0.80) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL15024639 0.89 LMNA (0.80) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL368130 0.88 LMNA (0.78) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL8432165 0.88 LMNA (0.78) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL14499615 0.88 LMNA (0.78) LMNATHRBCYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 14200 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026105121-A1 ANTICANCER FORMULATIONS AND USES THEREOF INTRAGEL THERAPEUTICS LTD. (IL) 2026-05-21 WO claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12570704-B2 Functionally modified maytansinoids and compositions and methods of use thereof University of Georgie Research Foundation, Inc. (US) 2026-03-10 US claimed
EP-4676551-A1 RADIATION SPACER HYDROGELS, METHODS OF FORMING, AND METHODS OF USE Clearstream Technologies Limited (IE) 2026-01-14 EP claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
EP-4524131-A1 SMALL MOLECULES FOR TREATING CANCER, INHABITING CHEMOKINE ACTIVITY AND/OR INDUCING CELL DEATH AlonBio Ltd. (IL) 2025-03-19 EP claimed
US-12202803-B2 Small molecules for treating cancer, inhibiting chemokine activity and/or inducing cell death ALONBIO LTD. (IL) 2025-01-21 US claimed
US-20240425752-A1 BILIRUBIN-COATED RADIO-LUMINESCENT PARTICLES PURDUE RESEARCH FOUNDATION (US) 2024-12-26 US claimed
EP-4086250-B1 MULTIFUNCTIONAL INHIBITORS OF MEK/PI3K AND MTOR/MEK/PI3K BIOLOGICAL PATHWAYS AND THERAPEUTIC METHODS USING THE SAME UNIV MICHIGAN REGENTS (US) 2024-12-11 EP claimed
US-20240343697-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2024-10-17 US claimed
CN-1261803-A Antioxidant enhancement of therapy for hyperproliferative conditions ATHEROGENICS INC (US) 2000-08-02 CN claimed
WO-2000043045-A1 METHOD FOR IMPROVED RADIATION THERAPY PHOTOGEN, INC. (US) 2000-07-27 WO claimed
WO-2000018439-A2 USE OF NEOANGIOGENESIS MARKERS FOR DIAGNOSING AND TREATING TUMOURS BY THERAPY SCHERING AKTIENGESELLSCHAFT (DE) 2000-04-06 WO claimed
WO-1999030693-A2 A DOUBLE CAPSULE FOR THE ADMINISTRATION OF ACTIVE PRINCIPLES IN MULTIPLE THERAPIES AXCAN PHARMA INC. (CA) 1999-06-24 WO claimed
WO-1999012548-A1 TREATMENT OF INFLAMMATORY CONDITIONS THERAMARK LIMITED (GB) 1999-03-18 WO claimed
US-5612310-A ANTITUMOR AGENTS AND NITRIC OXIDE SCAVENGERS, REDUCING BLOOD FLOW, HYPOXIC CYCLOTOXIN FOR CARDIOVASCULAR DISORDERS DUKE UNIVERSITY (US) 1997-03-18 US claimed
US-5554638-A ADMINISTERING NITRIC OXIDE SYNTHASE INHIBITOR AND HYPOXIC CYTOTOXIN DUKE UNIVERSITY (US) 1996-09-10 US claimed
US-5192784-A Physical and chemical stability DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-03-09 US claimed
EP-0359347-B1 COVALENTLY-LINKED COMPLEXES AND METHODS FOR ENHANCED CYTOTOXICITY AND IMAGING NEORX CORPORATION (US) 1992-12-23 EP claimed
EP-0287317-A2 Platinum complexes with one radiosensitizing ligand THE BRITISH COLUMBIA CANCER FOUNDATION (CA) 1988-10-19 EP claimed