SCHEMBL4414048

SCHEMBL4414048

C=C(F)C(F)(F)C([O])c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 3/20 0.40
SRC P12931 2/20 0.38
CES1 P23141 2/20 0.38
CES2 O00748 1/20 0.38
PTPN1 P18031 2/20 0.36
HPGD P15428 1/20 0.36
CYP2D6 P10635 1/20 0.35
LMNA P02545 2/20 0.34
MAPK1 P28482 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL382252 0.73 ACP3 (0.42) ACP3SRCCES1CES2PTPN1
SCHEMBL28258273 0.70 ACP3 (0.40) ACP3SRCCES1CES2PTPN1
SCHEMBL28088550 0.67 POLB (0.39) ACP3SRCCES1CES2PTPN1
SCHEMBL17956469 0.64 TSHR (0.43) SRCCES1CES2CYP2D6LMNA
SCHEMBL5042134 0.64 ATM (0.42) SRCCES1CES2CYP2D6
SCHEMBL17363627 0.64 HPGD (0.35) ACP3SRCHPGDCYP2D6LMNA
SCHEMBL28837273 0.63 SRC (0.39) ACP3SRCCES1CES2PTPN1
SCHEMBL4274555 0.63 SRC (0.39) ACP3SRCCES1CES2PTPN1
SCHEMBL29009915 0.63 CYP2D6 (0.43) ACP3SRCCES1CES2CYP2D6
SCHEMBL15114536 0.63 LMNA (0.47) ACP3SRCCES1CES2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009144548-A1 IMIDAZO [2,1-B] PURINE DERIVATIVES AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2009-12-03 WO disclosed