SCHEMBL4415013

SCHEMBL4415013

CC(C)CN[C@]1(N2CC[C@H](NC(=O)c3cccc(C(F)(F)F)c3)C2=O)CCCC[C@H]1CS(=O)(=O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 20/20 0.55
KCNH2 Q12809 4/20 0.55
CCR5 P51681 3/20 0.47
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4415012 0.86 CCR2 (0.61) CCR2KCNH2CCR5CYP2D6
SCHEMBL4421946 0.82 CCR2 (0.62) CCR2KCNH2CCR5
SCHEMBL4424621 0.80 CCR2 (0.54) CCR2KCNH2CCR5
SCHEMBL4415009 0.78 CCR2 (0.59) CCR2KCNH2CCR5CYP2D6
SCHEMBL4413543 0.77 CCR2 (0.55) CCR2KCNH2CCR5
SCHEMBL4417518 0.76 CCR2 (0.64) CCR2KCNH2CCR5CYP2D6
SCHEMBL4423202 0.75 CCR2 (0.66) CCR2KCNH2CCR5CYP2D6
SCHEMBL4416767 0.75 CCR2 (0.53) CCR2KCNH2CCR5
SCHEMBL4414936 0.74 CCR2 (0.57) CCR2KCNH2CCR5CYP2D6
SCHEMBL4415142 0.73 CCR2 (0.46) CCR2KCNH2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1606255-B1 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2009-11-11 EP claimed
EP-1606255-B1 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2009-11-11 EP disclosed