Amodiaquine

Amodiaquine

SCHEMBL44152

CCN(CC)Cc1cc(Nc2ccnc3cc(Cl)ccc23)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 9/20 1.00
CYP1A2 P05177 8/20 1.00
KCNH2 Q12809 5/20 1.00
APP P05067 5/20 1.00
NR4A2 P43354 2/20 1.00
ABCB11 O95342 1/20 1.00
CHRM2 P08172 1/20 1.00
HTR1A P08908 1/20 1.00
CHRM1 P11229 1/20 1.00
DRD2 P14416 1/20 1.00
ADRA2C P18825 1/20 1.00
SLC6A2 P23975 1/20 1.00
PTGS2 P35354 1/20 1.00
OPRM1 P35372 1/20 1.00
HTR2B P41595 1/20 1.00
CYP2J2 P51589 1/20 1.00
SLC6A3 Q01959 1/20 1.00
HRH3 Q9Y5N1 1/20 1.00
CYP2C8 P10632 6/20 0.98
CYP2C19 P33261 6/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Amodiaquine SCHEMBL29441086 1.00 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL29425350 1.00 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL317888 0.99 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL12094969 0.99 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL29430175 0.99 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL29788983 0.99 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL1491204 0.98 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL284774 0.98 CYP2D6 (0.96) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL30903900 0.98 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
SCHEMBL20536537 0.94 CYP2D6 (0.88) CYP2D6CYP1A2KCNH2APPNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8281 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4680248-A1 PRODUCTS OF MANUFACTURE AND THERAPEUTIC COMPOSITIONS FOR TREATING, AMELIORATING OR PREVENTING VIRAL INFECTIONS AND METHODS FOR MAKING AND USING THEM Topelia Aust Limited (ACN 652 771 670) (AU) 2026-01-21 EP claimed
EP-4680608-A1 2,6-DIHYDRO-7H-PYRAZOLO[3,4-C]PYRIDIN-7-ONE DERIVATIVES AS ANTI-MALARIAL AGENTS MMV Medicines for Malaria Venture (CH) 2026-01-21 EP claimed
EP-4677612-A1 METHODS FOR DETERMINING DRUG CANDIDATES mosaiques diagnostics & therapeutics AG (DE) 2026-01-14 EP claimed
US-12509439-B2 Anti-malarial agents UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2025-12-30 US claimed
US-20250388603-A1 ANTIMALARIAL COMPOUNDS SCRIPPS RESEARCH INST (US) 2025-12-25 US claimed
EP-4659817-A2 LIPOSOME COMPOSITION FOR USE IN PERITONEAL DIALYSIS Versantis AG (CH) 2025-12-10 EP claimed
WO-2025244856-A1 METHODS AND COMPOSITIONS RELATING TO ELQ COMPOUNDS OREGON HEALTH & SCIENCE UNIVERSITY (US) 2025-11-27 WO claimed
EP-3625238-B1 NOVEL SPIRO-LACTAM COMPOUNDS, PROCESS AND USES THEREOF UNIV DE COIMBRA (PT) 2025-11-26 EP claimed
US-12458694-B2 Methods for treatment of accelerated atherosclerosis and rheumatoid arthritis with an anti-Apo B100 antibody ABCENTRA, LLC (US) 2025-11-04 US claimed
EP-0338532-A2 N-alkylamino derivates of aromatic, tricyclic compounds in the treatment of drug-resistant protozoal infections MERRELL DOW PHARMACEUTICALS INC. (US) 1989-10-25 EP claimed
WO-1989008119-A1 HIGH MOLECULAR WEIGHT PRODRUG DERIVATIVES OF ANTI-INFLAMMATORY DRUGS SELCH LARSEN CLAUS (DK) 1989-09-08 WO claimed
EP-0331471-A1 High molecular weight prodrug derivatives of antiinflammatory drugs Larsen, Claus Selch (DK) 1989-09-06 EP claimed
US-4806537-A Use of amodiaquin and related compounds in treatment of nervous system degeneration CITY OF HOPE (US) 1989-02-21 US claimed
EP-0290959-A2 Drug mixture for prophylaxis and therapy of malaria HOECHST AKTIENGESELLSCHAFT (DE) 1988-11-17 EP claimed
EP-0037175-B1 PHARMACEUTICAL COMPOSITIONS EFAMOL LIMITED (GB) 1988-02-10 EP claimed
EP-0152379-A2 Process for preparing pharmaceutical compositions containing unilamellar liposomes CIBA-GEIGY AG (CH) 1985-08-21 EP claimed
EP-0035856-B1 PHARMACEUTICAL AND DIETARY COMPOSITIONS EFAMOL LIMITED (GB) 1984-07-04 EP claimed
EP-0037175-A1 Pharmaceutical compositions EFAMOL LIMITED (GB) 1981-10-07 EP claimed
EP-0035856-A2 Pharmaceutical and dietary compositions EFAMOL LIMITED (GB) 1981-09-16 EP claimed