Amodiaquine

Amodiaquine

SCHEMBL29425350

CCN(CC)Cc1cc(Nc2ccnc3cc(Cl)ccc23)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 9/20 1.00
CYP1A2 P05177 8/20 1.00
KCNH2 Q12809 5/20 1.00
APP P05067 5/20 1.00
NR4A2 P43354 2/20 1.00
ABCB11 O95342 1/20 1.00
CHRM2 P08172 1/20 1.00
HTR1A P08908 1/20 1.00
CHRM1 P11229 1/20 1.00
DRD2 P14416 1/20 1.00
ADRA2C P18825 1/20 1.00
SLC6A2 P23975 1/20 1.00
PTGS2 P35354 1/20 1.00
OPRM1 P35372 1/20 1.00
HTR2B P41595 1/20 1.00
CYP2J2 P51589 1/20 1.00
SLC6A3 Q01959 1/20 1.00
HRH3 Q9Y5N1 1/20 1.00
CYP2C8 P10632 6/20 0.98
CYP2C19 P33261 6/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Amodiaquine SCHEMBL29441086 1.00 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL44152 1.00 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL317888 0.99 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL12094969 0.99 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL29430175 0.99 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL29788983 0.99 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL1491204 0.98 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL284774 0.98 CYP2D6 (0.96) CYP2D6CYP1A2KCNH2APPNR4A2
Amodiaquine SCHEMBL30903900 0.98 CYP2D6 (1.00) CYP2D6CYP1A2KCNH2APPNR4A2
SCHEMBL20536537 0.94 CYP2D6 (0.88) CYP2D6CYP1A2KCNH2APPNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250269005-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT TOPELIA AUST LIMITED (ACN 652 771 670) (AU) 2025-08-28 US claimed
EP-4337179-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT Topelia Aust Limited (ACN 652 771 670) (AU) 2024-03-20 EP claimed
WO-2022236364-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT TOPELIA AUST LIMITED (ACN 652 771 670) (AU) 2022-11-17 WO claimed
WO-2022214855-A1 USE OF NITAZOXANIDE TO PREPARE A MEDICINAL PRODUCT TO PREVENT OR TREAT CORONAVIRUS SARS-COV-2 INFECTION SIEGFRIED RHEIN, S.A. DE C.V. (MX) 2022-10-13 WO claimed
CN-114118146-A Rolling bearing fault diagnosis method and system based on belief rule base 南京晨光集团有限责任公司 2022-03-01 CN claimed
CN-121574131-A Heterocyclic compounds for insect repellent 勃林格殷格翰动物保健有限公司 2026-02-27 CN disclosed
US-20250269005-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT TOPELIA AUST LIMITED (ACN 652 771 670) (AU) 2025-08-28 US disclosed
WO-2025133005-A1 IONISING RADIATION DETECTOR ELECTRICITE DE FRANCE (FR) 2025-06-26 WO disclosed
WO-2025052381-A1 INHIBITORS AND COMBINATIONS FOR TREATING DISEASES HADASIT MEDICAL RESEARCH SERVICES AND DEVELOPMENT LTD. (IL) 2025-03-13 WO disclosed
US-12233122-B2 Methods for treating, ameliorating or preventing infections using drug and vaccination combination treatment TOPELIA AUST LIMITED (652 771 670) (AU) 2025-02-25 US disclosed
US-20240382578-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT TOPELIA AUST LTD 652 771 670 (AU) 2024-11-21 US disclosed
EP-4337179-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT Topelia Aust Limited (ACN 652 771 670) (AU) 2024-03-20 EP disclosed
US-11857617-B2 Methods for treating, ameliorating or preventing infections using drug and vaccination combination treatment TOPELIA AUST LIMITED (652 771 670) (AU) 2024-01-02 US disclosed
CN-115947684-A Method for preparing 4-aminoquinoline derivatives through palladium and copper concerted catalytic oxidation aromatization 贵州医科大学 2023-04-11 CN disclosed
CN-115943307-A MR1 ligands and pharmaceutical compositions for immunomodulation 巴塞尔大学 2023-04-07 CN disclosed
US-20220370589-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT TOPELIA AUST LIMITED (ACN 652 771 670) (AU) 2022-11-24 US disclosed
WO-2022236364-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT TOPELIA AUST LIMITED (ACN 652 771 670) (AU) 2022-11-17 WO disclosed
WO-2022214855-A1 USE OF NITAZOXANIDE TO PREPARE A MEDICINAL PRODUCT TO PREVENT OR TREAT CORONAVIRUS SARS-COV-2 INFECTION SIEGFRIED RHEIN, S.A. DE C.V. (MX) 2022-10-13 WO disclosed
CN-114600329-A Method and apparatus for controlled switching of coupled loads 日立能源瑞士股份公司 2022-06-07 CN disclosed
CN-114118146-A Rolling bearing fault diagnosis method and system based on belief rule base 南京晨光集团有限责任公司 2022-03-01 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240382578-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT ACE, ACE2, CASP3 CYP2D6 390/4885CYP1A2 1177/4885KCNH2 1886/4885
US-12233122-B2 Methods for treating, ameliorating or preventing infections using drug and vaccination combination treatment ACE, ACE2, CASP3 CYP2D6 390/4885CYP1A2 1177/4885KCNH2 1886/4885
US-11857617-B2 Methods for treating, ameliorating or preventing infections using drug and vaccination combination treatment ZFX, IKZF3, ACE2 CYP2D6 1348/4885CYP1A2 1203/4885KCNH2 533/4885
US-20250269005-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT ZFX, ACE2, ZFR CYP2D6 1552/4885CYP1A2 1173/4885KCNH2 613/4885
US-20220370589-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT ZFX, IKZF3, ACE2 CYP2D6 1348/4885CYP1A2 1203/4885KCNH2 533/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.