SCHEMBL4418261

SCHEMBL4418261

COc1cc2c(c(OC)c1)C(c1cccc(OC(F)(F)F)c1)N(C(=O)c1cc(F)c(OC)c(F)c1F)CC2

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 1/20 0.41
GRIN2C Q14957 3/20 0.40
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
LMNA P02545 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
FKBP1A P62942 1/20 0.37
PPIB P23284 1/20 0.36
PPIA P62937 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
TP53 P04637 1/20 0.36
ABCB1 P08183 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4424502 0.87 NPSR1 (0.43) MTNR1BGRIN2CKMT2AMEN1LMNA
SCHEMBL4423047 0.85 GRIN2C (0.51) MTNR1BGRIN2CKMT2AMEN1LMNA
SCHEMBL4418256 0.84 KMT2A (0.52) GRIN2CKMT2AMEN1LMNANPSR1
SCHEMBL4416192 0.84 GRIN2C (0.47) MTNR1BGRIN2CKMT2AMEN1LMNA
SCHEMBL4413447 0.84 KMT2A (0.55) GRIN2CKMT2AMEN1LMNANPSR1
SCHEMBL4417027 0.84 MTNR1B (0.47) MTNR1BGRIN2CKMT2AMEN1LMNA
SCHEMBL4418264 0.84 MTNR1B (0.52) MTNR1BGRIN2CKMT2AMEN1LMNA
SCHEMBL6509279 0.82 GRIN2C (0.52) MTNR1BGRIN2CKMT2AMEN1LMNA
SCHEMBL4416759 0.81 GRIN2C (0.53) GRIN2CKMT2AMEN1LMNANPSR1
SCHEMBL4414983 0.81 GRIN2C (0.43) MTNR1BGRIN2CKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663983-B1 N-SUBSTITUTED, 6,8-DIALKOXY-1,2,3,4-TETRAHYDRO-1H-ISOQUINOLINE AS POTASSIUM CHANNELS MODULATORS 4SC AG (DE) 2009-01-21 EP disclosed