SCHEMBL4420767

SCHEMBL4420767

CCOc1cc(C(=O)N2CCC3(CC2)CC(=O)c2c[c]ccc2O3)cc(OC)c1-c1cnn(C)c1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ACACB O00763 12/20 0.48
ACACA Q13085 1/20 0.43
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL730528 0.89 ACACB (0.52) ACACBACACAKMT2A
SCHEMBL4417682 0.85 ACACB (0.49) ACACBACACAKMT2A
SCHEMBL742140 0.85 ACACB (0.49) ACACBACACAKMT2A
SCHEMBL741079 0.84 ACACB (0.53) ACACBACACA
SCHEMBL730518 0.84 ACACB (0.47) ACACBACACAKMT2A
SCHEMBL731214 0.84 ACACB (0.53) ACACBACACA
SCHEMBL733394 0.84 ACACB (0.63) ACACBACACAKMT2A
SCHEMBL731131 0.84 ACACB (0.47) ACACBACACAKMT2A
SCHEMBL730697 0.84 ACACB (0.47) ACACBACACAKMT2A
SCHEMBL733228 0.83 ACACB (0.46) ACACBACACAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP claimed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO claimed
EP-2120569-B1 SPIROCHROMANON DERIVATIVES MERCK SHARP & DOHME (US) 2013-08-14 EP disclosed