SCHEMBL4425276

SCHEMBL4425276

CC(=O)On1ccc2c(O)cccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.42
HTR6 P50406 1/20 0.42
NOTUM Q6P988 2/20 0.38
THRB P10828 1/20 0.37
BAZ2B Q9UIF8 1/20 0.36
BAZ2A Q9UIF9 1/20 0.36
CA12 O43570 3/20 0.35
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA7 P43166 3/20 0.35
CA9 Q16790 3/20 0.35
CA14 Q9ULX7 3/20 0.35
CYP3A4 P08684 1/20 0.35
POLB P06746 1/20 0.34
MAPT P10636 2/20 0.34
HTT P42858 1/20 0.34
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16493596 0.82 NOTUM (0.37) HTR6NOTUMCYP3A4POLBMAPT
SCHEMBL27771802 0.81 HTR2C (0.41) HTR2CHTR6CA12CA1CA2
SCHEMBL4949214 0.79 HTR2C (0.46) HTR2CHTR6NOTUMTHRBCA12
SCHEMBL11217145 0.78 NR4A2 (0.47) THRBMAPTGAALMNAMEN1
SCHEMBL1716468 0.78 POLB (0.43) POLBMAPTHTTGAALMNA
SCHEMBL4417523 0.77 GAA (0.44) THRBPOLBMAPTGAAMEN1
SCHEMBL27807548 0.77 POLB (0.42) POLBMAPTHTTGAALMNA
SCHEMBL28576274 0.77 POLB (0.42) POLBMAPTHTTGAALMNA
SCHEMBL4954033 0.75 HTR2C (0.43) HTR2CHTR6THRBCA12CA1
SCHEMBL4955621 0.75 HTR2C (0.46) HTR2CHTR6THRBCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094662-A1 POLYCYCLIC ACID COMPOUNDS USEFUL AS CRTH2 ANTAGONISTS AND ANTIALLERGIC AGENTS Astellas Pharma Inc. (JP) 2009-09-02 EP disclosed
WO-2008072784-A1 POLYCYCLIC ACID COMPOUNDS USEFUL AS CRTH2 ANTAGONISTS AND ANTIALLERGIC AGENTS ASTELLAS PHARMA INC. (JP) 2008-06-19 WO disclosed