SCHEMBL4428657

SCHEMBL4428657

COc1ccc2cccc(C(CN3CCC(NC(=O)OC(C)(C)C)CC3)C(=O)O)c2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.44
MTNR1B P49286 2/20 0.44
KCNA3 P22001 1/20 0.44
CKS1B P61024 1/20 0.41
SKP1 P63208 1/20 0.41
SKP2 Q13309 1/20 0.41
CCR5 P51681 1/20 0.40
PARP1 P09874 2/20 0.40
DRD2 P14416 4/20 0.39
SLC2A1 P11166 2/20 0.39
DRD3 P35462 1/20 0.38
PDE10A Q9Y233 1/20 0.38
KDM4D Q6B0I6 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
OGFRL1 Q5TC84 1/20 0.36
USP14 P54578 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3209072 0.93 MTNR1A (0.44) MTNR1AMTNR1BKCNA3CKS1BSKP1
SCHEMBL4477066 0.90 SLC2A1 (0.46) MTNR1AMTNR1BKCNA3CKS1BSKP1
SCHEMBL3154477 0.88 MTNR1A (0.44) MTNR1AMTNR1BKCNA3CKS1BSKP1
SCHEMBL4491260 0.80 MTNR1A (0.47) MTNR1AMTNR1BKCNA3CKS1BSKP1
SCHEMBL3148938 0.80 SLC2A1 (0.41) MTNR1AMTNR1BKCNA3CKS1BSKP1
SCHEMBL3551289 0.80 SLC2A1 (0.51) KCNA3SLC2A1KDM4D
SCHEMBL3144945 0.80 KCNA3 (0.40) MTNR1AMTNR1BKCNA3CKS1BSKP1
SCHEMBL5726714 0.78 SLC2A1 (0.61) SLC2A1
SCHEMBL3155389 0.78 MTNR1A (0.48) MTNR1AMTNR1BSLC2A1
SCHEMBL1267791 0.77 SLC2A1 (0.40) MTNR1AMTNR1BKCNA3CKS1BSKP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136807-A1 PYRROLO (3, 2, 1-IJ) QUINOLINE-4-ONE DERIVATIVES FOR TREATING TUBERCULOSIS Glaxo Group Limited (GB) 2009-12-30 EP disclosed
WO-2008125594-A1 PYRROLO (3, 2, 1-IJ) QUINOLINE-4-ONE DERIVATIVES FOR TREATING TUBERCULOSIS GLAXO GROUP LIMITED (GB) 2008-10-23 WO disclosed