SCHEMBL4428953

SCHEMBL4428953

CCC(C)(c1ccc(OCC(O)C(C)(C)C)c(C)c1)c1cc(C)cs1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
VDR P11473 11/20 0.60
AR P10275 4/20 0.57
HDAC6 Q9UBN7 8/20 0.54
HDAC3 O15379 4/20 0.54
HDAC1 Q13547 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3395694 0.90 VDR (0.64) VDRARHDAC6HDAC3HDAC1
SCHEMBL6437088 0.80 HDAC6 (0.53) VDRARHDAC6HDAC3HDAC1
SCHEMBL16183084 0.77 VDR (0.77) VDRARHDAC6HDAC3HDAC1
SCHEMBL13366805 0.74 HDAC6 (0.66) VDRARHDAC6HDAC3HDAC1
SCHEMBL20059951 0.74 VDR (0.60) VDRARHDAC6HDAC3HDAC1
SCHEMBL15076968 0.73 VDR (0.75) VDRARHDAC6HDAC3HDAC1
SCHEMBL2949160 0.73 VDR (0.75) VDRARHDAC6HDAC3HDAC1
SCHEMBL16178018 0.73 VDR (0.75) VDRARHDAC6HDAC3HDAC1
Lg-190178 SCHEMBL29754199 0.72 VDR (1.00) VDRAR
SCHEMBL2946827 0.72 VDR (0.73) VDRARHDAC6HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1511740-B1 PHENYL-THIOPHENE TYPE VITAMIN D RECEPTOR MODULATORS LILLY CO ELI (US) 2009-07-08 EP disclosed