SCHEMBL4429372

SCHEMBL4429372

NC(=O)CC(c1ccc(Cl)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.51
PPARG P37231 4/20 0.47
PPARA Q07869 1/20 0.47
UTS2R Q9UKP6 4/20 0.45
CACNA1A O00555 1/20 0.44
CACNA2D1 P54289 1/20 0.44
CACNA1B Q00975 1/20 0.44
CACNB1 Q02641 1/20 0.44
CACNA1C Q13936 1/20 0.44
GABBR2 O75899 3/20 0.44
GABBR1 Q9UBS5 3/20 0.44
CYP2C9 P11712 3/20 0.44
LMNA P02545 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CYP3A4 P08684 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
NFKB1 P19838 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438449 0.87 CACNA1A (0.56) CNR2CACNA1ACACNA2D1CACNA1BCACNB1
SCHEMBL4617540 0.87 CYP2C19 (0.55) CACNA1ACACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL4431819 0.84 CYP2C19 (0.55) CNR2UTS2RCACNA1ACACNA2D1CACNA1B
SCHEMBL4441848 0.81 CACNA1A (0.57) PPARGCACNA1ACACNA2D1CACNB1CYP2C9
SCHEMBL10955012 0.80 TACR1 (0.59) CNR2UTS2RLMNARHOCRHOA
SCHEMBL1980002 0.79 KMT2A (0.55) PPARGPPARAGABBR2GABBR1CYP2C9
SCHEMBL11080075 0.78 CES2 (0.47) CNR2
SCHEMBL7485566 0.78 FFAR1 (0.56) CNR2PPARGCACNA1ACACNA2D1CACNA1B
SCHEMBL4432755 0.77 AKR1C3 (0.51) PPARGPPARACACNA1ACACNA2D1CACNB1
SCHEMBL23080122 0.77 CES2 (0.50) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed