SCHEMBL4429386

SCHEMBL4429386

CNC(=O)[C@H](NCC[C@@H](c1ccc(C(F)(F)F)cc1)c1ccccc1OC)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.44
MEN1 O00255 4/20 0.44
OPRM1 P35372 2/20 0.44
OPRD1 P41143 1/20 0.44
KDM4E B2RXH2 2/20 0.43
CCR2 P41597 3/20 0.42
ALDH1A1 P00352 3/20 0.41
LMNA P02545 2/20 0.41
HTT P42858 2/20 0.41
MITF O75030 1/20 0.41
MAPT P10636 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
MTTP P55157 2/20 0.40
BLM P54132 1/20 0.40
CCR3 P51677 1/20 0.40
CNR1 P21554 2/20 0.39
NPC1 O15118 2/20 0.39
CYP2D6 P10635 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4436216 1.00 KMT2A (0.44) KMT2AMEN1OPRM1OPRD1KDM4E
SCHEMBL4438661 0.89 KDM4E (0.45) KMT2AMEN1KDM4ECCR2ALDH1A1
SCHEMBL4440273 0.89 KDM4E (0.45) KMT2AMEN1KDM4ECCR2ALDH1A1
SCHEMBL4436222 0.88 KDM4E (0.40) KMT2AMEN1OPRM1KDM4ECCR2
SCHEMBL4435280 0.88 KDM4E (0.40) KMT2AMEN1OPRM1KDM4ECCR2
SCHEMBL4433693 0.88 KDM4E (0.49) KMT2AMEN1OPRM1KDM4ECCR2
SCHEMBL4431735 0.88 KDM4E (0.49) KMT2AMEN1OPRM1KDM4ECCR2
SCHEMBL4432373 0.88 KDM4E (0.43) KMT2AMEN1OPRD1KDM4ECCR2
SCHEMBL4429519 0.88 KDM4E (0.43) KMT2AMEN1OPRD1KDM4ECCR2
SCHEMBL4440275 0.88 KDM4E (0.44) KMT2AMEN1OPRM1KDM4ECCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed