SCHEMBL4435280

SCHEMBL4435280

CNC(=O)[C@H](NCC[C@@H](c1ccc(C(F)(F)F)cc1)c1cccnc1OC)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
CCR2 P41597 6/20 0.39
ALDH1A1 P00352 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
EP300 Q09472 3/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
P2RY1 P47900 1/20 0.37
CNR1 P21554 2/20 0.37
NPC1 O15118 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C19 P33261 2/20 0.37
MTOR P42345 2/20 0.37
RAB9A P51151 2/20 0.37
CNR2 P34972 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4436222 1.00 KDM4E (0.40) KDM4ECCR2ALDH1A1CTDSP1HCRTR1
SCHEMBL4430416 0.89 CNR1 (0.48) ALDH1A1SLC6A2SLC6A4EP300GAA
SCHEMBL4432975 0.89 CNR1 (0.48) ALDH1A1SLC6A2SLC6A4EP300GAA
SCHEMBL4436216 0.88 KMT2A (0.44) KDM4ECCR2ALDH1A1CTDSP1HCRTR1
SCHEMBL4429386 0.88 KMT2A (0.44) KDM4ECCR2ALDH1A1CTDSP1HCRTR1
SCHEMBL4438661 0.85 KDM4E (0.45) KDM4ECCR2ALDH1A1CTDSP1EP300
SCHEMBL4440273 0.85 KDM4E (0.45) KDM4ECCR2ALDH1A1CTDSP1EP300
SCHEMBL4433693 0.85 KDM4E (0.49) KDM4ECCR2ALDH1A1CTDSP1SLC6A2
SCHEMBL4431735 0.85 KDM4E (0.49) KDM4ECCR2ALDH1A1CTDSP1SLC6A2
SCHEMBL4434954 0.84 CNR1 (0.54) KDM4EALDH1A1SLC6A2SLC6A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed