SCHEMBL443014

SCHEMBL443014

NC(=O)Oc1cccc(F)c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.73
MEN1 O00255 2/20 0.73
PARP1 P09874 1/20 0.52
ESR1 P03372 1/20 0.51
ESR2 Q92731 1/20 0.51
KCNN4 O15554 4/20 0.47
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
PPARG P37231 1/20 0.45
PPARA Q07869 1/20 0.45
MAOB P27338 1/20 0.44
PARP10 Q53GL7 1/20 0.44
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
KCNH2 Q12809 1/20 0.43
SCN3A Q9NY46 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28147531 0.98 KMT2A (0.70) KMT2AMEN1PARP1ESR1ESR2
Methylene Chloride SCHEMBL27910646 0.93 KMT2A (0.63) KMT2AMEN1PARP1ESR1ESR2
SCHEMBL5487011 0.83 ESR1 (0.54) KMT2AMEN1PARP1ESR1ESR2
SCHEMBL17004183 0.82 ESR1 (0.53) KMT2AMEN1PARP1ESR1ESR2
SCHEMBL18697278 0.82 ESR1 (0.53) KMT2AMEN1PARP1ESR1ESR2
SCHEMBL5580391 0.80 ESR1 (0.51) KMT2AMEN1PARP1ESR1ESR2
SCHEMBL287805 0.80 CYP3A4 (0.63) KMT2AMEN1ESR1ESR2MAOB
SCHEMBL6987573 0.79 MEN1 (0.50) KMT2AMEN1PARP1ESR1ESR2
SCHEMBL442239 0.79 MEN1 (0.52) KMT2AMEN1PARP1CES2CES1
SCHEMBL28783426 0.78 KMT2A (0.53) KMT2AMEN1PARP1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 91 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113214339-A Panaxadiol derivatives, preparation method and medical application thereof 延边大学 2021-08-06 CN claimed
CN-106749074-A A kind of preparation method of Fang oxazolidinones intermediate 沈阳药科大学 2017-05-31 CN claimed
CN-105849366-A Method and composition for hydraulic fracturing and for tracing oil production 光谱追踪服务有限公司 2016-08-10 CN claimed
CN-103443099-A Compositions and methods for modulating FXR IRM LLC 2013-12-11 CN claimed
CN-102985417-A Piperidin-4-yl azetidine derivatives as JAK1 inhibitors INCYTE CORP 2013-03-20 CN claimed
CN-101166733-A Pyrazole derivatives as phosphodiesterase 4 inhibitors MEMORY PHARM CORP (US) 2008-04-23 CN claimed
CN-101056628-A Ester derivatives and medicinal use thereof JAPAN TOBACCO INC (JP) 2007-10-17 CN claimed
CN-117500786-A TEAD inhibitors 奥赖恩公司 2024-02-02 CN disclosed
CN-113683629-B Substituted heteroaryl compounds, compositions and uses thereof 北京范恩柯尔生物科技有限公司 2023-07-04 CN disclosed
CN-108976222-B Heterocyclic ring-containing biaryl oxazolidinone compound and preparation method thereof 沈阳药科大学 2021-09-03 CN disclosed
CN-113214339-A Panaxadiol derivatives, preparation method and medical application thereof 延边大学 2021-08-06 CN disclosed
CN-105120860-B Histone deacetylase inhibitors 生物马林药物股份有限公司 2021-01-26 CN disclosed
CN-109111451-A Dihydropyrimidines and its application in drug 广东东阳光药业有限公司 2019-01-01 CN disclosed
CN-1646125-A Substituted pyridones as modulators of P38MAP kinase PHARMACIA CORP (US) 2005-07-27 CN disclosed
CN-1646426-A Metallized mesoporous silicate and method of oxidation with the same SUMITOMO CHEMICAL CO (JP) 2005-07-27 CN disclosed
WO-2004077511-A2 (METH)ACRYLIC AND (METH)ACRYLAMIDE MONOMERS, POLYMERIZABLE COMPOSITIONS, AND POLYMERS OBTAINED THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2004-09-10 WO disclosed
CN-1432014-A Triazole compound of amide series SANKYO CO (JP) 2003-07-23 CN disclosed
EP-1062207-A1 9-AMINOACRIDINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Samjin Pharmaceutical Co., Ltd. (KR) 2000-12-27 EP disclosed
WO-2000037447-A1 9-AMINOACRIDINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-06-29 WO disclosed
CN-1152306-A Process for preparing 5-aryl-2, 4-dialkyl-3H-1, 2, 4-triazole-3-thiones MERRELL PHARMA INC (US) 1997-06-18 CN disclosed