SCHEMBL4430306

SCHEMBL4430306

NC(=O)C(CC1CCN(CCc2ccccc2)C1)(c1ccccc1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 4/20 0.55
CHRM2 P08172 2/20 0.50
CCR3 P51677 1/20 0.49
HTR2A P28223 2/20 0.47
ADRB2 P07550 1/20 0.47
CHRM4 P08173 1/20 0.47
ADRB1 P08588 1/20 0.47
CHRM5 P08912 1/20 0.47
ADRA2A P08913 1/20 0.47
CHRM1 P11229 1/20 0.47
DRD2 P14416 1/20 0.47
KCNE1 P15382 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
HRH2 P25021 1/20 0.47
SLC6A4 P31645 1/20 0.47
ADRA1A P35348 1/20 0.47
OPRM1 P35372 1/20 0.47
OPRK1 P41145 1/20 0.47
HTR2B P41595 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8879133 0.93 CHRM3 (0.57) CHRM3CCR3HTR2ASIGMAR1
SCHEMBL8878260 0.83 CHRM3 (0.56) CHRM3CCR3
Water SCHEMBL10720338 0.80 BCHE (0.51) CHRM3
SCHEMBL9361492 0.79 CHRM3 (0.69) CHRM3CHRM2HTR2AADRB2CHRM4
SCHEMBL9361499 0.79 CHRM3 (0.69) CHRM3CHRM2HTR2AADRB2CHRM4
SCHEMBL6630519 0.77 CCR3 (0.59) CCR3HTR2ALTA4HSIGMAR1
SCHEMBL6628169 0.77 CCR3 (0.59) CCR3HTR2ALTA4HSIGMAR1
SCHEMBL11023730 0.75 CCR3 (0.64) CCR3SIGMAR1
SCHEMBL843343 0.75 CCR3 (0.64) CCR3HTR2A
SCHEMBL7465330 0.75 CCR3 (0.64) CCR3HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121594-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2009-11-25 EP disclosed
WO-2008103426-A1 QUATERNARY AMMONIUM DIPHENYLMETHYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2008-08-28 WO disclosed