SCHEMBL8878260

SCHEMBL8878260

NC(=O)C(CC1CCN(Cc2ccccc2)CC1)(c1ccccc1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 3/20 0.56
GAA P10253 1/20 0.56
ACHE P22303 5/20 0.55
BCHE P06276 2/20 0.55
CCR3 P51677 1/20 0.52
CXCR4 P61073 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8879133 0.87 CHRM3 (0.57) CHRM3ACHECCR3
Water SCHEMBL10720338 0.84 BCHE (0.51) CHRM3ACHEBCHE
SCHEMBL4430306 0.83 CHRM3 (0.55) CHRM3CCR3
SCHEMBL4757520 0.80 CHRM3 (0.48) CHRM3
SCHEMBL10519952 0.79 CCR3 (0.59) CHRM3ACHEBCHECCR3CXCR4
SCHEMBL4756802 0.79 CHRM3 (0.47) CHRM3
SCHEMBL9248078 0.78 KMT2A (0.57) CCR3
SCHEMBL26096555 0.78 ACHE (0.72) GAAACHEBCHECCR3
SCHEMBL1138416 0.77 ACHE (0.76) CHRM3ACHEBCHECCR3
SCHEMBL4854037 0.77 GAA (0.64) GAAACHEBCHECCR3CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607950-A IRRITABLE BOWEL SYNDROME PFIZER INC. (US) 1997-03-04 US disclosed
EP-0508988-B1 MUSCARINIC RECEPTOR ANTAGONISTS PFIZER LTD (GB) 1994-03-02 EP disclosed
WO-1991010647-A1 MUSCARINIC RECEPTOR ANTAGONISTS PFIZER LIMITED (GB) 1991-07-25 WO disclosed