Bicarbonate

Bicarbonate

SCHEMBL4432364

COc1ccc(CC(=O)NC2CCC(C)CC2)c(Cl)c1.O=C(O)O

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
GAA P10253 1/20 0.56
SIGMAR1 Q99720 6/20 0.50
LMNA P02545 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPK1 P28482 1/20 0.47
EPHX2 P34913 1/20 0.47
KDM4E B2RXH2 1/20 0.47
SMYD3 Q9H7B4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL4428400 0.90 MEN1 (0.70) MEN1KMT2ASIGMAR1SMN1; SMN2EPHX2
Bicarbonate SCHEMBL4433306 0.89 MEN1 (0.56) MEN1KMT2AGAASIGMAR1EPHX2
Bicarbonate SCHEMBL4428116 0.89 MEN1 (0.56) MEN1KMT2AGAASIGMAR1SMN1; SMN2
Bicarbonate SCHEMBL4428096 0.89 KMT2A (0.72) MEN1KMT2ASIGMAR1SMN1; SMN2EPHX2
Bicarbonate SCHEMBL4434715 0.89 KMT2A (0.72) MEN1KMT2ASIGMAR1SMN1; SMN2EPHX2
Bicarbonate SCHEMBL4434731 0.88 MEN1 (0.55) MEN1KMT2AGAASIGMAR1EPHX2
Bicarbonate SCHEMBL4424931 0.87 MEN1 (0.54) MEN1KMT2AGAASIGMAR1SMN1; SMN2
Bicarbonate SCHEMBL4435168 0.87 MEN1 (0.51) MEN1KMT2AGAASIGMAR1EPHX2
Bicarbonate SCHEMBL6996704 0.87 MEN1 (0.58) MEN1KMT2AGAASIGMAR1LMNA
Bicarbonate SCHEMBL4425148 0.86 MEN1 (0.56) MEN1KMT2AGAASIGMAR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741700-B1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER CROPSCIENCE AG (DE) 2009-10-07 EP disclosed
EP-0741700-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AG (DE) 1996-11-13 EP disclosed
WO-1995020572-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1995-08-03 WO disclosed