Bicarbonate

Bicarbonate

SCHEMBL4428096

COc1ccc(CC(=O)NC2CCCCC2)c(Cl)c1.O=C(O)O

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.72
MEN1 O00255 3/20 0.72
EPHX2 P34913 1/20 0.61
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2C19 P33261 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
HPGD P15428 1/20 0.55
MAPT P10636 1/20 0.54
POLB P06746 2/20 0.52
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.48
USP2 O75604 1/20 0.48
HTT P42858 1/20 0.48
ALDH1A1 P00352 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL4434715 1.00 KMT2A (0.72) KMT2AMEN1EPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL4428400 0.99 MEN1 (0.70) KMT2AMEN1EPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL4432364 0.89 MEN1 (0.57) KMT2AMEN1EPHX2SMN1; SMN2SIGMAR1
Bicarbonate SCHEMBL4428116 0.88 MEN1 (0.56) KMT2AMEN1EPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL4433306 0.88 MEN1 (0.56) KMT2AMEN1EPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL4425148 0.88 MEN1 (0.56) KMT2AMEN1EPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL4434731 0.87 MEN1 (0.55) KMT2AMEN1EPHX2SIGMAR1ALDH1A1
Bicarbonate SCHEMBL6996071 0.86 MEN1 (0.73) KMT2AMEN1EPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL6992780 0.86 MEN1 (0.73) KMT2AMEN1EPHX2CYP1A2CYP3A4
Bicarbonate SCHEMBL4424931 0.86 MEN1 (0.54) KMT2AMEN1EPHX2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741700-B1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER CROPSCIENCE AG (DE) 2009-10-07 EP disclosed
EP-0741700-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AG (DE) 1996-11-13 EP disclosed
WO-1995020572-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1995-08-03 WO disclosed