SCHEMBL4432457

SCHEMBL4432457

CC(=O)C(c1ccc(F)c(C)c1)c1cnc(C)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
RAB9A P51151 3/20 0.39
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
S1PR3 Q99500 4/20 0.34
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33
AKT1 P31749 1/20 0.33
ALDH1A1 P00352 2/20 0.33
PIM1 P11309 1/20 0.33
MMP13 P45452 1/20 0.33
GAA P10253 1/20 0.33
S1PR1 P21453 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438585 0.87 S1PR3 (0.42) S1PR3KCNQ3KCNQ2S1PR1
SCHEMBL4431484 0.84 APLNR (0.38) S1PR3HDAC3HDAC1HDAC2HDAC6
SCHEMBL4433750 0.83 HDAC4 (0.35) NPC1RAB9ALMNAHDAC3HDAC1
SCHEMBL4433370 0.80 PDE2A (0.40) SMN1; SMN2LMNAHDAC3HDAC1HDAC2
SCHEMBL4441500 0.80 AKR1C3 (0.34) SMN1; SMN2MAPTS1PR3AKR1C3AKR1C2
SCHEMBL4441218 0.77 PDE4A (0.41) GRIN2B
SCHEMBL4434008 0.76 AKR1C3 (0.39) HDAC3HDAC1HDAC2HDAC6AKR1C3
SCHEMBL4435119 0.76 KCNQ3 (0.41) S1PR3HDAC3HDAC1HDAC2HDAC6
SCHEMBL4440506 0.75 AKR1C3 (0.38) NPC1SMN1; SMN2RAB9ALMNAMAPT
SCHEMBL4440986 0.74 BRD4 (0.46) S1PR3AKR1C3AKR1C2S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed