SCHEMBL4432901

SCHEMBL4432901

CNC(=O)[C@H](NCC[C@H](c1ccc(C(F)(F)F)cc1)c1ccc(OC(C)C)c(OC(C)C)c1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
CCR2 P41597 5/20 0.41
ALDH1A1 P00352 2/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
ALOX5 P09917 3/20 0.40
EPHX2 P34913 3/20 0.40
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
LMNA P02545 4/20 0.39
NPC1 O15118 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 2/20 0.39
MTOR P42345 2/20 0.39
RAB9A P51151 2/20 0.39
CYP3A4 P08684 2/20 0.39
SLC6A2 P23975 2/20 0.39
HTR2C P28335 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4434528 0.95 KMT2A (0.43) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4429248 0.95 KMT2A (0.43) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4433516 0.95 KMT2A (0.43) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4433201 0.95 KMT2A (0.43) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4434762 0.93 PDE4A (0.42) KDM4ECCR2ALDH1A1CTDSP1MEN1
SCHEMBL4429756 0.93 PDE4A (0.42) KDM4ECCR2ALDH1A1CTDSP1MEN1
SCHEMBL4429519 0.89 KDM4E (0.43) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4432373 0.89 KDM4E (0.43) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4431735 0.87 KDM4E (0.49) KDM4ECCR2ALDH1A1CTDSP1ALOX5
SCHEMBL4433693 0.87 KDM4E (0.49) KDM4ECCR2ALDH1A1CTDSP1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed