SCHEMBL4433692

SCHEMBL4433692

COc1ccc(CC(N)(CN)Cc2ccc(OC)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.53
MAOB P27338 3/20 0.48
IDO1 P14902 4/20 0.48
AGXT P21549 2/20 0.48
TDP1 Q9NUW8 2/20 0.46
MAPK1 P28482 1/20 0.46
SLC6A4 P31645 1/20 0.46
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 2/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
LTA4H P09960 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
AOC3 Q16853 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5514194 0.84 IDO1 (0.48) TAAR1MAOBIDO1AGXTTDP1
SCHEMBL9583292 0.82 TAAR1 (0.52) TAAR1MAOBIDO1AGXTTDP1
SCHEMBL8621821 0.80 CYP19A1 (0.47) TAAR1IDO1AGXTMAPK1ALDH1A1
SCHEMBL27990275 0.79 TAAR1 (0.48) TAAR1MAOBIDO1AGXTTDP1
SCHEMBL183751 0.79 SLC6A2 (0.57) TAAR1MAOBIDO1AGXTTDP1
SCHEMBL27715705 0.78 IDO1 (0.45) TAAR1MAOBIDO1AGXTALDH1A1
Hydrochloric Acid SCHEMBL3800374 0.78 SLC6A2 (0.55) TAAR1MAOBIDO1AGXTTDP1
SCHEMBL11336433 0.78 IDO1 (0.50) TAAR1MAOBIDO1AGXTTDP1
SCHEMBL23458084 0.77 TAAR1 (0.48) TAAR1IDO1AGXTTDP1SLC6A4
SCHEMBL9583891 0.77 TAAR1 (0.46) TAAR1MAOBIDO1AGXTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4069418-A1 PROCESS FOR PREPARING AMINES OVER A COPPER CATALYST BASF SE (DE) 2022-10-12 EP disclosed
WO-2021110472-A1 PROCESS FOR PREPARING AMINES OVER A COPPER CATALYST BASF SE (DE) 2021-06-10 WO disclosed
EP-2114899-A2 CONTROLLED RELEASE OF ACTIVE ALDEHYDES AND KETONES FROM EQUILIBRATED DYNAMIC MIXTURES Firmenich S.A. (CH) 2009-11-11 EP disclosed
WO-2008093272-A2 CONTROLLED RELEASE OF ACTIVE ALDEHYDES AND KETONES FROM EQUILIBRATED DYNAMIC MIXTURES FIRMENICH SA (CH) 2008-08-07 WO disclosed
EP-1765833-A2 NEWS SALTS IN THE PREPARATION OF CEPHALOSPORIN ANTIBIOTICS Orchid Chemicals and Pharmaceuticals Limited (IN) 2007-03-28 EP disclosed
WO-2006006040-A2 NEWS DIAMINE SALTS OF CEPHALOSPORIN ANTIBIOTICS AND THEIR PREPARATION ORCHID CHEMICALS & PHARMACEUTICALS LIMITED (IN) 2006-01-19 WO disclosed