SCHEMBL4433778

SCHEMBL4433778

O=C(c1csc(-c2cc[c]cc2)n1)N1CCOCC1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.61
PIN1 Q13526 1/20 0.47
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.44
CNR1 P21554 1/20 0.44
RAB9A P51151 7/20 0.44
NPC1 O15118 6/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP1A2 P05177 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2104945 0.85 HTR2C (0.45) HTR2CALDH1A1KDM4EHPGDRAB9A
SCHEMBL3543512 0.79 IRAK4 (0.64) HTR2CALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL3541979 0.77 HTR2C (0.56) HTR2CALDH1A1KDM4EHPGDRAB9A
SCHEMBL31206570 0.75 HTR2C (0.58) HTR2CHPGDRAB9ANPC1SMN1; SMN2
SCHEMBL4398770 0.74 PIN1 (0.44) HTR2CPIN1ALDH1A1HPGDRAB9A
SCHEMBL26707398 0.74 HPGD (0.61) HTR2CHPGDCNR1RAB9ANPC1
SCHEMBL3545567 0.73 HTR2C (0.67) HTR2CHPGDCNR1RAB9ANPC1
SCHEMBL2225857 0.73 HDAC1 (0.55) HTR2CPIN1
SCHEMBL3543198 0.73 HTR2C (0.63) HTR2CPIN1ALDH1A1KDM4EHPGD
SCHEMBL29944217 0.73 HTR2C (0.63) HTR2CPIN1ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504413-B2 N-(4-(imidazo[1,2A]pyridin-YL)phenethyl)benzamide inhibitors of the mitotic kinesin CENP-E for treating certain cellular proliferation diseases CYTOKINETICS, INC. (US) 2009-03-17 US disclosed
CN-101023057-A Certain chemicals, compositions, and methods CYTOKINETICS INC (US) 2007-08-22 CN disclosed