SCHEMBL4434611

SCHEMBL4434611

CNC(=O)[C@H](NCC[C@@H](c1ccc(C(F)(F)F)nc1)c1ccc(F)c(OC)c1)c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 10/20 0.41
EPHX2 P34913 3/20 0.38
MAPK1 P28482 2/20 0.38
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CYP2J2 P51589 1/20 0.37
NTRK1 P04629 1/20 0.36
CSF1R P07333 1/20 0.36
NTRK2 Q16620 1/20 0.36
KCNK3 O14649 1/20 0.36
ROCK2 O75116 1/20 0.35
TACR1 P25103 1/20 0.35
CCR2 P41597 1/20 0.35
EP300 Q09472 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441204 1.00 P2RX7 (0.41) P2RX7EPHX2MAPK1CYP2C9CYP2C19
SCHEMBL4438596 0.95 P2RX7 (0.41) P2RX7KCNK3EP300
SCHEMBL4433559 0.95 P2RX7 (0.41) P2RX7KCNK3EP300
SCHEMBL4432133 0.94 P2RX7 (0.41) P2RX7ROCK2EP300
SCHEMBL4432125 0.94 P2RX7 (0.41) P2RX7ROCK2EP300
SCHEMBL4441632 0.93 P2RX7 (0.41) P2RX7EPHX2MAPK1CYP2C9CYP2C19
SCHEMBL4435140 0.92 P2RX7 (0.40) P2RX7EPHX2MAPK1CYP2C9CYP2C19
SCHEMBL4429693 0.91 P2RX7 (0.45) P2RX7EPHX2MAPK1CYP2C9CYP2C19
SCHEMBL4428035 0.91 P2RX7 (0.45) P2RX7EPHX2MAPK1CYP2C9CYP2C19
SCHEMBL4440233 0.90 PDE4A (0.42) P2RX7NTRK1CSF1RNTRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed