SCHEMBL4435240

SCHEMBL4435240

CNC(=O)[C@H](NCC[C@@H](c1ccc(Cl)cc1)c1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.50
ALDH1A1 P00352 4/20 0.48
CTDSP1 Q9GZU7 1/20 0.48
CASR P41180 2/20 0.46
KDM4E B2RXH2 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CCR2 P41597 3/20 0.44
KLRK1 P26718 1/20 0.44
MICA Q29983 1/20 0.44
RAET1L Q5VY80 1/20 0.44
CNR2 P34972 2/20 0.44
UTS2R Q9UKP6 3/20 0.43
EP300 Q09472 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4436339 1.00 CNR1 (0.50) CNR1ALDH1A1CTDSP1CASRKDM4E
SCHEMBL4433693 0.94 KDM4E (0.49) CNR1ALDH1A1CTDSP1KDM4ESMN1; SMN2
SCHEMBL4431735 0.94 KDM4E (0.49) CNR1ALDH1A1CTDSP1KDM4ESMN1; SMN2
SCHEMBL4441758 0.92 ALDH1A1 (0.47) CNR1ALDH1A1CTDSP1CASRKDM4E
SCHEMBL4441724 0.92 ALDH1A1 (0.47) CNR1ALDH1A1CTDSP1CASRKDM4E
SCHEMBL4436364 0.91 ALDH1A1 (0.48) CNR1ALDH1A1CTDSP1CASRKDM4E
SCHEMBL4429569 0.91 ALDH1A1 (0.48) CNR1ALDH1A1CTDSP1CASRKDM4E
SCHEMBL4427927 0.90 CNR1 (0.51) CNR1ALDH1A1CTDSP1CASRKDM4E
SCHEMBL4434552 0.90 CNR1 (0.51) CNR1ALDH1A1CTDSP1CASRKDM4E
SCHEMBL4441777 0.89 KDM4E (0.46) ALDH1A1CTDSP1KDM4ESMN1; SMN2CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed