SCHEMBL4435780

SCHEMBL4435780

CNC(=O)[C@H](NCC[C@H](c1ccc(Cl)nc1)c1ccc(OC(F)F)c(OC(F)F)c1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 19/20 0.43
KCNH2 Q12809 2/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
HTR1E P28566 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
S1PR3 Q99500 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441767 0.90 PDE4A (0.41) PDE4AKCNH2MEN1ALDH1A1LMNA
SCHEMBL4429537 0.88 PDE4A (0.47) PDE4AKCNH2
SCHEMBL4429160 0.86 PDE4A (0.43) PDE4AMEN1ALDH1A1LMNATP53
SCHEMBL4429325 0.86 PDE4A (0.43) PDE4AMEN1ALDH1A1LMNATP53
SCHEMBL4434957 0.83 PDE4A (0.42) PDE4AKCNH2MEN1ALDH1A1LMNA
SCHEMBL4429756 0.83 PDE4A (0.42) PDE4AKCNH2MEN1ALDH1A1LMNA
SCHEMBL4434762 0.83 PDE4A (0.42) PDE4AKCNH2MEN1ALDH1A1LMNA
SCHEMBL4438606 0.81 PDE4A (0.42) PDE4AKCNH2ALDH1A1
SCHEMBL4429658 0.81 PDE4A (0.41) PDE4AKCNH2
SCHEMBL4441413 0.81 PDE4A (0.41) PDE4AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed