SCHEMBL4437511

SCHEMBL4437511

NCCc1nc2cccc(Cl)c2nc1-c1cccc(F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 7/20 0.43
ADORA2A P29274 4/20 0.41
DPP4 P27487 2/20 0.39
NT5E P21589 1/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
ADORA1 P30542 3/20 0.36
ADORA2B P29275 1/20 0.34
MAP4K4 O95819 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
HRH1 P35367 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4185412 0.90 DPP4 (0.43) TAAR1ADORA2ADPP4NT5EMEN1
SCHEMBL27802876 0.88 ADORA2A (0.39) ADORA2ADPP4NT5EMEN1USP2
SCHEMBL4441851 0.88 ADORA2A (0.39) ADORA2ADPP4NT5EMEN1USP2
SCHEMBL4171148 0.85 ERBB2 (0.42) ADORA2ADPP4NT5EMEN1USP2
SCHEMBL4431468 0.84 TAAR1 (0.36) TAAR1DPP4CYP1A2CYP3A4CYP2C9
SCHEMBL14047509 0.81 ADORA2A (0.38) ADORA2ADPP4NT5EMEN1USP2
SCHEMBL4182457 0.78 NR1H2 (0.51) ADORA2ANT5EMEN1USP2ALDH1A1
SCHEMBL16447644 0.77 ADORA2A (0.39) ADORA2ADPP4NT5EMEN1USP2
SCHEMBL4172215 0.76 SMN1; SMN2 (0.43) ADORA2AMEN1USP2ALDH1A1CYP1A2
SCHEMBL4431751 0.76 MAP4K4 (0.41) MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137186-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES Amgen Inc. (US) 2009-12-30 EP disclosed
WO-2008118468-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2008-10-02 WO disclosed