SCHEMBL4437810

SCHEMBL4437810

Cc1ccc(NCCCCNS(=O)(=O)c2ccccc2[N+](=O)[O-])c(C)c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
MAPT P10636 2/20 0.54
HTT P42858 2/20 0.54
KAT2B Q92831 3/20 0.52
NPY5R Q15761 3/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP19A1 P11511 1/20 0.49
F13A1 P00488 1/20 0.48
TGM1 P22735 1/20 0.48
GAA P10253 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31284709 0.82 KMT2A (0.68) ALDH1A1HTTNPY5RMEN1KMT2A
SCHEMBL13763409 0.81 ALDH1A1 (0.52) ALDH1A1MAPTHTTNPY5RMEN1
SCHEMBL3540913 0.80 KMT2A (0.66) ALDH1A1HTTNPY5RMEN1KMT2A
SCHEMBL27006685 0.79 KMT2A (0.68) ALDH1A1HTTNPY5RMEN1KMT2A
SCHEMBL29571128 0.79 KMT2A (0.68) ALDH1A1HTTNPY5RMEN1KMT2A
SCHEMBL4067677 0.78 KMT2A (0.60) ALDH1A1HTTNPY5RMEN1KMT2A
SCHEMBL3228138 0.78 SMN1; SMN2 (0.45) ALDH1A1MAPTHTTMEN1KMT2A
SCHEMBL3228129 0.78 SMN1; SMN2 (0.45) ALDH1A1MAPTHTTMEN1KMT2A
SCHEMBL14572299 0.77 RECQL (0.62) ALDH1A1HTTNPY5RMEN1KMT2A
SCHEMBL14572312 0.77 RECQL (0.62) ALDH1A1HTTNPY5RMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136811-A1 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF Boehringer Ingelheim International GmbH (DE) 2009-12-30 EP disclosed
WO-2008124745-A1 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-10-16 WO disclosed