SCHEMBL4439247

SCHEMBL4439247

c1nnn(Cc2ccsc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.37
HTR1A P08908 1/20 0.36
HTR2C P28335 1/20 0.36
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
KDM4A O75164 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
S1PR1 P21453 1/20 0.31
CYP17A1 P05093 1/20 0.31
CYP11B1 P15538 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3116533 0.68 CYP19A1 (0.58) TAAR1HTR1AALDH1A1MEN1KDM4A
SCHEMBL2351887 0.67 CYP19A1 (0.64) CYP11B1CYP11B2
SCHEMBL31272207 0.67 POLB (0.40) HTR1AHTR2CALDH1A1MEN1MAPT
SCHEMBL2563333 0.66 TAAR1 (0.43) TAAR1ADORA3ADORA2AADORA2BADORA1
SCHEMBL4834371 0.65 CYP19A1 (0.48) ALDH1A1MEN1MAPTKMT2AL3MBTL1
SCHEMBL1491120 0.63 KDM4E (0.59) TAAR1ADORA3ADORA2AADORA2BADORA1
SCHEMBL4701933 0.62 ALDH1A1 (0.48) TAAR1ALDH1A1KMT2ADRD2DRD3
SCHEMBL10674754 0.62 HRH3 (0.56) ALDH1A1L3MBTL1OPRM1OPRD1OPRK1
SCHEMBL8671494 0.61 TAAR1 (0.71) TAAR1ADORA2AALDH1A1MEN1KDM4A
SCHEMBL9369371 0.61 CYP11B1 (0.61) MAPTCYP17A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097410-A1 HETEROARYL-PYRAZOLE DERIVATIVES AS CANNABINOID CB1 RECEPTOR ANTAGONISTS Green Cross Corporation (KR) 2009-09-09 EP claimed
WO-2008039023-A1 HETEROARYL-PYRAZOLE DERIVATIVES AS CANNABINOID CB1 RECEPTOR ANTAGONISTS GREEN CROSS CORPORATION (KR) 2008-04-03 WO claimed