SCHEMBL4440640

SCHEMBL4440640

COC(=O)[C@H](Cc1ccc(C(F)(F)F)nc1)NC(=O)[C@@H](C)N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.44
CYP2C19 P33261 3/20 0.44
ALDH1A1 P00352 2/20 0.44
THRB P10828 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TSHR P16473 2/20 0.42
NOS3 P29474 3/20 0.41
NOS1 P29475 3/20 0.41
NOS2 P35228 3/20 0.41
IL1RN P18510 2/20 0.41
ERAP2 Q6P179 2/20 0.41
ERAP1 Q9NZ08 1/20 0.41
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40
KCNQ4 P56696 1/20 0.40
KCNQ5 Q9NR82 1/20 0.40
CYP2D6 P10635 2/20 0.39
CYP2C8 P10632 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4447526 0.88 MME (0.44) CA2
SCHEMBL18256473 0.82 KLK5 (0.47) NOS3NOS1NOS2KCNQ3KCNQ2
SCHEMBL1519828 0.82 KLK5 (0.47) NOS3NOS1NOS2KCNQ3KCNQ2
SCHEMBL1519826 0.82 KLK5 (0.47) NOS3NOS1NOS2KCNQ3KCNQ2
SCHEMBL4445933 0.82 ALDH1A1 (0.45) CYP2C9CYP2C19ALDH1A1KCNQ3KCNQ2
SCHEMBL13323761 0.79 KLK5 (0.42)
SCHEMBL4448480 0.79 ALDH1A1 (0.53) CYP2C9CYP2C19ALDH1A1TSHRCYP2D6
Trifluoroacetic Acid SCHEMBL16461603 0.77 ALDH1A1 (0.51) CYP2C9CYP2C19ALDH1A1THRBHSD17B10
SCHEMBL13755248 0.76 TSHR (0.65) CYP2C9CYP2C19ALDH1A1THRBHSD17B10
SCHEMBL27543181 0.76 ALDH1A1 (0.56) CYP2C9CYP2C19ALDH1A1THRBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531507-B2 Acylated nonadepsipeptides containing pyridyl alanine residues AICURIS GMBH & CO. KG (DE) 2009-05-12 US disclosed