SCHEMBL4441012

SCHEMBL4441012

COc1cncc(Br)c1.COc1cncc(N)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MKNK2 Q9HBH9 2/20 0.38
ROCK2 O75116 1/20 0.38
MAP4K4 O95819 1/20 0.38
PRKACA P17612 1/20 0.38
ROCK1 Q13464 1/20 0.38
DYRK1A Q13627 1/20 0.38
NTRK3 Q16288 1/20 0.38
PKN2 Q16513 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
STK17A Q9UEE5 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
MKNK1 Q9BUB5 1/20 0.37
CYP1A1 P04798 1/20 0.37
CYP1B1 Q16678 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31162408 0.88
SCHEMBL113446 0.88
SCHEMBL7444 0.88
SCHEMBL3881071 0.86 CYP1A1 (0.43) CYP3A4MKNK2ROCK2MAP4K4PRKACA
Bromide SCHEMBL4761808 0.86 ALDH1A1 (0.45) CYP3A4ALDH1A1MKNK2ROCK2MAP4K4
Hydrochloric Acid SCHEMBL3933926 0.86 ALDH1A1 (0.45) CYP3A4ALDH1A1MKNK2ROCK2MAP4K4
Cyanide SCHEMBL28133661 0.82 CYP1A1 (0.41) CYP3A4MKNK2ROCK2MAP4K4PRKACA
Formic Acid SCHEMBL28134510 0.78 MKNK2 (0.41) MKNK2ROCK2MAP4K4PRKACAROCK1
SCHEMBL116722 0.77
SCHEMBL5848746 0.76 CYP1A1 (0.47) ALDH1A1CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137177-A2 AURORA KINASE MODULATORS AND METHOD OF USE Amgen, Inc (US) 2009-12-30 EP disclosed
WO-2008124083-A2 AURORA KINASE MODULATORS AND METHOD OF USE AMGEN INC. (US) 2008-10-16 WO disclosed