SCHEMBL4441702

SCHEMBL4441702

CNC(=O)[C@@H](NCC[C@@H](c1ccc(OC)cc1)c1ccc(C(F)(F)F)nc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.48
KMT2A Q03164 7/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
MITF O75030 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
CASR P41180 2/20 0.45
P2RX7 Q99572 7/20 0.44
EP300 Q09472 1/20 0.42
MEN1 O00255 4/20 0.42
BLM P54132 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CRHBP P24387 1/20 0.41
CYP2C19 P33261 1/20 0.41
CRHR2 Q13324 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4433971 1.00 CNR1 (0.48) CNR1CNR2KMT2ALMNAHTT
SCHEMBL4434777 0.89 KMT2A (0.39) CNR1CNR2KMT2ALMNAHTT
SCHEMBL4430291 0.88 P2RX7 (0.41) ALDH1A1P2RX7EP300
SCHEMBL4434565 0.88 P2RX7 (0.41) ALDH1A1P2RX7EP300
Hydrochloric Acid SCHEMBL4432260 0.87 P2RX7 (0.41) KMT2AALDH1A1P2RX7EP300MEN1
SCHEMBL4433559 0.87 P2RX7 (0.41) KMT2AALDH1A1P2RX7EP300
SCHEMBL4438596 0.87 P2RX7 (0.41) KMT2AALDH1A1P2RX7EP300
SCHEMBL4432377 0.87 P2RX7 (0.40) KMT2AALDH1A1P2RX7EP300
SCHEMBL4431769 0.87 P2RX7 (0.40) KMT2AALDH1A1P2RX7EP300
SCHEMBL4434954 0.86 CNR1 (0.54) CNR1CNR2KMT2ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed