SCHEMBL4443019

SCHEMBL4443019

Nc1ncc(-c2cccc(C(=O)NCCCN3CCOCC3)c2)nc1-c1nc2ccccc2[nH]1

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATR Q13535 14/20 0.69
MAP4K4 O95819 1/20 0.53
GRK5 P34947 1/20 0.51
POLB P06746 2/20 0.51
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
MAPK1 P28482 1/20 0.51
DUSP3 P51452 1/20 0.51
PTPN5 P54829 1/20 0.51
PTPN11 Q06124 1/20 0.51
KMT2A Q03164 1/20 0.49
MAPK8 P45983 1/20 0.48
MAPK10 P53779 1/20 0.48
MAPK14 Q16539 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4013029 0.95 ATR (0.73) ATRMAP4K4GRK5KDM4EALDH1A1
SCHEMBL4455054 0.92 ATR (0.76) ATRMAP4K4
SCHEMBL4014260 0.92 ATR (0.68) ATR
SCHEMBL4163487 0.92 ATR (0.68) ATR
SCHEMBL4450649 0.83 ATR (0.68) ATR
SCHEMBL4443884 0.83 ATR (0.70) ATR
SCHEMBL3063607 0.82 ATR (1.00) ATR
SCHEMBL29458584 0.82 ATR (1.00) ATR
SCHEMBL2481992 0.80 ATR (1.00) ATR
SCHEMBL4010962 0.80 ATR (0.68) ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO claimed