Daunorubicin

Daunorubicin

SCHEMBL4444

COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(C)=O)C[C@@H]3O[C@H]1C[C@H](N)[C@H](O)[C@H](C)O1.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TOP2A

The experimentally established mechanism targets of Daunorubicin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A known ✓ P11388 5/20 0.99
MEN1 O00255 10/20 1.00
THRB P10828 10/20 1.00
KMT2A Q03164 10/20 1.00
BLM P54132 9/20 1.00
RECQL P46063 8/20 1.00
SMN1; SMN2 Q16637 7/20 1.00
MAPT P10636 7/20 1.00
BRCA1 P38398 6/20 1.00
HIF1A Q16665 6/20 1.00
USP2 O75604 5/20 1.00
S100A4 P26447 5/20 1.00
MAPK1 P28482 5/20 1.00
CYP3A4 P08684 4/20 1.00
NPC1 O15118 4/20 1.00
RAB9A P51151 4/20 1.00
PAX8 Q06710 3/20 1.00
POLB P06746 3/20 1.00
HSP90AA1 P07900 2/20 1.00
HSP90AB1 P08238 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Daunorubicin SCHEMBL31326687 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL142541 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL31725676 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL4445 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL122984 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL4659664 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL20185623 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL2217102 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL20204237 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL
Daunorubicin SCHEMBL29462666 1.00 MEN1 (1.00) MEN1THRBKMT2ABLMRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 27345 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260132141-A1 PROTEIN PHOSPHATASE 2A ACTIVATORS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2026-05-14 US claimed
EP-3856736-B1 NOVEL COMPOUNDS AS NADPH OXIDASE INHIBITORS CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2026-05-06 EP claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
EP-3969123-B1 LYMPHOTOXIN ALPHA FOR USE IN THERAPY OF MYELOID LEUKEMIA CYCURIA THERAPEUTICS GMBH (AT) 2026-04-29 EP claimed
US-20260109699-A1 AZOLE DERIVATIVES AS SHP2 INHIBITORS IRBM S.P.A. (IT) 2026-04-23 US claimed
EP-4727933-A1 COMBINATION THERAPY METHODS FOR TREATING TP53-Y220C MUTANT AND TP53 WILDTYPE LEUKEMIAS Board of Regents, The University of Texas System (US) 2026-04-22 EP claimed
US-20260102373-A1 LYMPH DIRECTING PRODRUGS MONASH UNIVERSITY (AU) 2026-04-16 US claimed
US-20260096569-A1 EDIBLE COATING WITH ANTIMICROBIAL PROPERTIES APEEL TECH INC (US) 2026-04-09 US claimed
EP-4709378-A1 COMPOUNDS FOR NOS-RELATED CANCERS AND METHODS OF USE Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. (IL) 2026-03-18 EP claimed
US-20260069700-A1 BRUSH PRODRUGS AND USES THEREOF MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2026-03-12 US claimed
EP-0580171-A2 Pharmaceutical composition containing a carrier bound antitumor substance KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1994-01-26 EP claimed
EP-0525073-A1 ANTHRAQUINONES AS INHIBITORS OF SULFIDE PRODUCTION FROM SULFATE-REDUCING BACTERIA. DU PONT (US) 1993-02-03 EP claimed
EP-0088695-B1 ANTIBODY CONJUGATES CYTOGEN CORPORATION (US) 1992-06-03 EP claimed
EP-0306541-B1 PROCESS FOR OBTAINING DAUNORUBICIN-HYDROCHLORIDE FROM FERMENTATION BROTHS BIOGAL GYOGYSZERGYAR (HU) 1992-01-08 EP claimed
WO-1991015954-A1 ANTHRAQUINONES AS INHIBITORS OF SULFIDE PRODUCTION FROM SULFATE-REDUCING BACTERIA E.I. DU PONT DE NEMOURS AND COMPANY (US) 1991-10-31 WO claimed
US-5061492-A biodegeadeable polymer matrix is copolymer of gylcolic acid a nd lactic acid TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-10-29 US claimed
US-4925662-A ANTITUMOR AGENT BONDED TO HUMAN IMMUNOGLOBULIN KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1990-05-15 US claimed
US-4711782-A Prolonged release microcapsules and their production TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1987-12-08 US claimed
US-4671958-A Antibody conjugates for the delivery of compounds to target sites CYTOGEN CORPORATION (US) 1987-06-09 US claimed
EP-0122132-A2 Anti-tumour substance KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1984-10-17 EP claimed