SCHEMBL4444154

SCHEMBL4444154

OC1CC2CCC(C1)N2CCCN1c2ccccc2Sc2ccc(Cl)cc21

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.85
RAD52 P43351 4/20 0.85
KIF11 P52732 2/20 0.85
MAPT P10636 6/20 0.60
DRD2 P14416 5/20 0.60
CYP2C19 P33261 5/20 0.60
LMNA P02545 5/20 0.60
SMN1; SMN2 Q16637 5/20 0.60
MAPK1 P28482 5/20 0.60
ADRA2A P08913 4/20 0.60
ADRA2B P18089 4/20 0.60
ADRA2C P18825 4/20 0.60
SLC6A2 P23975 4/20 0.60
HTR2A P28223 4/20 0.60
HTR2C P28335 4/20 0.60
SLC6A4 P31645 4/20 0.60
HRH1 P35367 4/20 0.60
DRD3 P35462 4/20 0.60
HTR2B P41595 4/20 0.60
CYP1A2 P05177 4/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11244507 1.00 CYP2D6 (0.85) CYP2D6RAD52KIF11MAPTDRD2
SCHEMBL11246700 0.85 CYP2D6 (0.67) CYP2D6RAD52KIF11MAPTDRD2
SCHEMBL11237819 0.82 CYP2D6 (0.63) CYP2D6RAD52KIF11MAPTDRD2
SCHEMBL11244510 0.81 RAD52 (0.66) CYP2D6RAD52KIF11MAPTDRD2
SCHEMBL11237816 0.78 CYP2D6 (0.61) CYP2D6RAD52KIF11MAPTDRD2
SCHEMBL11244145 0.77 CYP2D6 (0.57) CYP2D6RAD52KIF11MAPTDRD2
SCHEMBL29724166 0.76 CYP2D6 (0.71) CYP2D6RAD52MAPTDRD2CYP2C19
SCHEMBL8053156 0.76 CYP2D6 (0.71) CYP2D6RAD52MAPTDRD2CYP2C19
SCHEMBL20412086 0.75 CYP2D6 (0.69) CYP2D6RAD52MAPTDRD2CYP2C19
SCHEMBL31673776 0.75 CYP2D6 (0.69) CYP2D6RAD52MAPTDRD2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8193238-B2 Inhibition of microtubule protrusion in cancer cells UNIVERSITY OF MARYLAND, BALTIMORE (US) 2012-06-05 US disclosed
US-20090137473-A1 INHIBITION OF MICROTUBULE PROTRUSION IN CANCER CELLS UNIVERSITY OF MARYLAND, BALTIMORE 2009-05-28 US disclosed
US-4366154-A TRANQUILIZERS; PSYCHOLOGICAL DISORDERS SANDOZ, INC. (US) 1982-12-28 US disclosed