Bromide

Bromide

SCHEMBL4445136

Br.Br.Br.Br.N=C(N)SCc1cccc(CSC(=N)N)c1-c1c(CSC(=N)N)cccc1CSC(=N)N

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.62
HPGD P15428 1/20 0.62
IDO1 P14902 10/20 0.61
TAAR1 Q96RJ0 3/20 0.61
LMNA P02545 3/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
SLC11A2 P49281 2/20 0.61
NOS1 P29475 2/20 0.56
NOS3 P29474 1/20 0.55
NOS2 P35228 1/20 0.55
MAPT P10636 1/20 0.52
ATP1A1 P05023 1/20 0.50
ATP1B1 P05026 1/20 0.50
ATP1A3 P13637 1/20 0.50
ATP1B2 P14415 1/20 0.50
ATP1A2 P50993 1/20 0.50
ATP1B3 P54709 1/20 0.50
FXYD2 P54710 1/20 0.50
ATP1A4 Q13733 1/20 0.50
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3690551 0.98 HTT (0.65) HTTHPGDIDO1TAAR1LMNA
Bromide SCHEMBL4018130 0.90 HTT (0.57) HTTHPGDIDO1TAAR1LMNA
Bromide SCHEMBL3686933 0.89 MAPT (0.59) HTTHPGDIDO1TAAR1LMNA
SCHEMBL3684767 0.88 HTT (0.59) HTTHPGDIDO1TAAR1LMNA
Bromide SCHEMBL2810146 0.87 IDO1 (0.71) HTTHPGDIDO1TAAR1LMNA
Bromide SCHEMBL4016347 0.87 NOS1 (0.60) HTTHPGDIDO1TAAR1LMNA
SCHEMBL14068776 0.86 MAPT (0.61) HTTHPGDIDO1TAAR1LMNA
SCHEMBL3691297 0.85 NOS1 (0.62) HTTHPGDIDO1TAAR1LMNA
SCHEMBL2812696 0.85 IDO1 (0.74) HTTHPGDIDO1TAAR1LMNA
Bromide SCHEMBL4017471 0.84 HTT (0.51) HTTHPGDIDO1TAAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061754-A1 BIARYL AND BIHETEROARYL COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2009-05-27 EP disclosed
WO-2008115999-A1 BIARYL AND BIHETEROARYL COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-09-25 WO disclosed